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PKC(蛋白激酶C)

PKC (protein kinase C) is a serine/threonine protein kinase that mediates insulin signaling, actin cytoskeleton, cell mobility, apoptosis and tumorigenesis etc.

Products for  PKC

  1. Cat.No. 产品名称 Information
  2. GC30545 Malantide Malantide是一种十二肽,能够被PKA磷酸化,并且能够增强PKA的活性。
  3. GC30200 PKC-theta inhibitor PKC-theta inhibitor (compound 20) inhibits PKC-θ with an IC50 of 18 nM.
  4. GC18521 Cercosporin A cytotoxic phytotoxin
  5. GC18354 Bisindolylmaleimide X (hydrochloride) A PKC inhibitor
  6. GC18246 R-59-949 A DGK-α inhibitor
  7. GC14134 1,2-Dimyristoyl-sn-glycerol A long-chain DAG
  8. GC18062 1,2-Dilauroyl-sn-glycerol A long-chain DAG
  9. GC12662 1,2-Distearoyl-sn-glycerol A diacylglycerol
  10. GC10299 Hexadecyl Methyl Glycerol A synthetic DAG
  11. GC16678 UCN-02 A PKC inhibitor
  12. GC13877 1,2-Dipalmitoyl-sn-glycerol A diacylglycerol
  13. GC17815 L-threo-Sphingosine C-18 A D-erythro-sphingosine analog
  14. GC13226 Bisindolylmaleimide VIII (acetate) A PKC inhibitor
  15. GC14716 Bisindolylmaleimide IV A PKC inhibitor
  16. GC10343 α-Amyloid Precursor Protein Modulator α-Amyloid Precursor Protein Modulator 是一种细胞可渗透的苯并内酰胺衍生蛋白激酶 C (PKC) 激活剂,Ki 为 11.9 nM。
  17. GC15018 Hispidin A polyphenol with diverse biological activities
  18. GC16405 Safingol A dual inhibitor of PKC and SPHK
  19. GC11022 SB 218078 A potent Chk1 inhibitor
  20. GC13273 ZIP ZIP 是 PKMζ 的选择性肽抑制剂。
  21. GC17239 Bisindolylmaleimide V A S6K inhibitor
  22. GC10029 Ro 31-8220 methanesulfonate Inhibitor of protein kinase C
  23. GC17242 (-)-epigallocatechin A green tea polyphenol
  24. GC10603 (-)-epicatechin gallate A natural polyphenol with diverse protective actions
  25. GC12695 Bryostatin 3 Bryostatin 3 是一种大环内酯,是一种蛋白激酶 C 激活剂,Ki 为 2.75 nM。 Bryostatin 3 可以阻断 12-O-tetradecanoylphorbol-13-acetate (TPA) 对细胞增殖的抑制作用,但不能阻断 TPA 增强的细胞-基质粘附。
  26. GC12842 Bryostatin 2 Protein kinase C (PKC) activator
  27. GC16475 Afuresertib A pan-Akt inhibitor
  28. GC14012 (-)-Indolactam V A PKC activator
  29. GC10682 TAS 301 An inhibitor of Ca2+ mobilization and CaM kinase II
  30. GC12135 Bisindolylmaleimide II A PKC inhibitor
  31. GC14583 R 59-022 A DGK inhibitor
  32. GC10820 Rottlerin An inhibitor of PKCδ and other protein kinases
  33. GC11605 C-1 C-1 是一种有效的蛋白激酶抑制剂,IC50 为 4 μM, 8 μM, 12 μM 和 240 μM 用于 cGMP 依赖性蛋白激酶 (PKG)、cAMP 依赖性蛋白激酶 (PKA) ,分别为蛋白激酶 C (PKC) 和 MLC 激酶。 C-1 也用作 ROCK 抑制剂。
  34. GC18055 SC-9 An activator of PKC
  35. GC13320 SC-10 Protein kinase C activator
  36. GC16510 ZIP, Biotinylated ZIP with a biotin moiety covalently attached
  37. GC15345 [Ala113]-MBP (104-118) [Ala113]-MBP (104-118) 是一种蛋白激酶 C (PKC) 的非竞争性肽抑制剂,IC50 范围为 28-62 μM。
  38. GC17727 [Ala107]-MBP (104-118) [Ala107]-MBP (104-118) 是一种蛋白激酶 C (PKC) 的非竞争性肽抑制剂,IC50 范围为 46-145 μM。
  39. GC11671 PKC fragment (530-558) Potent activator of protein kinase C
  40. GC15471 PKC β pseudosubstrate Selective cell-permeable peptide inhibitor of protein kinase C
  41. GC10404 PKC ζ pseudosubstrate PKC ζ pseudosubstrate 是一种选择性的细胞渗透性 PKC 抑制剂。
  42. GC11803 Pseudo RACK1 Activator of protein kinase C
  43. GC15148 Ionomycin calcium salt Ionomycin calcium salt是一种窄谱抗生素,对革兰氏阳性菌具有活性,由丛生链霉菌(Streptomyces conglobatus)产生。伊诺霉素钙盐可促进细胞凋亡。伊诺霉素还能诱导激活蛋白激酶 C (PKC)。.
  44. GC17563 LY 333531 hydrochloride A PKCβ inhibitor
  45. GC17352 Phorbol 12,13-dibutyrate An activator of PKC
  46. GC12027 FR 236924 An activator of PKCε
  47. GC10687 CGP 53353 CGP 53353 (DAPH-7) 是一种有效的 PKC 抑制剂,对 PKCβII 和 PKCβI 的 IC50 分别为 0.41 mM 和 3.8 mM。
  48. GC17670 Bryostatin 1 A marine macrolide with diverse biological activities
  49. GC15446 Ionomycin free acid A calcium ionophore
  50. GC11362 K 252a A non-selective PKC inhibitor
  51. GC11159 Calphostin C A selective PKC inhibitor

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