Home >> Signaling Pathways >> Tyrosine Kinase >> FGFR


FGFRs (fibroblast growth factor receptors) are transmembrane tyrosine kinase receptor. It is involved in carcinogenesis and plays an important role in cell differentiation, survival and proliferation etc.

  1. Cat.No. 产品名称 Information
  2. GC65516 Bemarituzumab
  3. GC65515 Aprutumab
  4. GC65212 FGFR1/DDR2 inhibitor 1 FGFR1/DDR2 inhibitor 1 is an inhibitor of fibroblast growth factor receptor 1 (FGFR1) and discoidin domain receptor 2 (DDR2).
  5. GC65179 MAX-40279
  6. GC64950 ODM-203 A dual inhibitor of VEGFR and FGFR
  7. GC64875 Gunagratinib
  8. GC64475 FGFR2-IN-2
  9. GC49700 Takeda-6d A dual inhibitor of RAF kinases and VEGFR2
  10. GC49686 N-desmethyl Regorafenib N-oxide An active metabolite of regorafenib
  11. GC63395 FGFR-IN-1
  12. GC62696 E7090 succinate
  13. GC62675 SM1-71
  14. GC62602 FGFR4-IN-5
  15. GC62291 (Z)-Orantinib
  16. GC62274 CPL304110
  17. GC61957 SU4984
  18. GC60726 CP-547632 TFA A potent inhibitor of VEGFR2 and bFGF
  19. GC50051 FIIN 1 hydrochloride FIIN 1 hydrochloride 是一种有效的、不可逆的、选择性的 FGFR 抑制剂。 FIIN 1 hydrochloride 与 FGFR1/2/3/4 和 Flt1/4 结合,Kd 分别为 2.8/6.9/5.4/120 nM 和 32/120 nM。 FIIN 1 hydrochloride 对 FGFR1/2/3/4 的生化 IC50 分别为 9.2、6.2、11.9 和 189 nM。
  20. GC45828 Ponatinib-d8 An internal standard for the quantification of ponatinib
  21. GC38575 CP-547632 hydrochloride A potent inhibitor of VEGFR2 and bFGF
  22. GC37773 TG 100801 Hydrochloride
  23. GC37772 TG 100572 Hydrochloride
  24. GC37771 TG 100572
  25. GC37679 SSR128129E free acid An FGFR inhibitor
  26. GC36745 Nintedanib esylate

    Nintedanib esylate, as a kinase inhibitor, used for the treatment of non-small cell lung cancer suffered from first-pass metabolism which resulted in low oral bioavailability .

  27. GC36546 Masitinib mesylate An inhibitor of c-Kit
  28. GC36438 Lenvatinib mesylate An inhibitor of VEGFR2 and VEGFR3
  29. GC36044 FIIN-3 An inhibitor of FGFRs
  30. GC44583 PD 089828 An inhibitor of EGFR, PDGFβ, FGF, and c-Src
  31. GC34476 ASP5878 ASP5878 is a novel FGFR-selective inhibitor with IC50 values of 0.47, 0.60, 0.74, and 3.5 nmol/L for recombinant FGFR1, 2, 3, and 4, respectively.
  32. GC34067 Rogaratinib (BAY1163877)
  33. GC34026 Tyrosine kinase-IN-1
  34. GC33519 2,5-Dihydroxybenzoic acid A benzoic acid with diverse biological activities
  35. GC33352 CP-547632 A potent inhibitor of VEGFR2 and bFGF
  36. GC32915 Pemigatinib An FGFR inhibitor
  37. GC32835 PP58
  38. GC32805 Sulfatinib (HMPL-012) A multi-kinase inhibitor
  39. GC32802 PRN1371 An irreversible pan-FGFR inhibitor
  40. GC32760 Dovitinib lactate (CHIR-258 lactate) A multi-kinase inhibitor
  41. GC32127 Alofanib (RPT835) An allosteric inhibitor of FGFR2
  42. GC31495 PF-05231023 A bioconjugation linker
  43. GC30767 Heparan Sulfate


  44. GC19399 Derazantinib An inhibitor of FGFR
  45. GC19341 SUN11602 An FGF2 mimetic
  46. GC19317 S49076 S49076 是一种新型、有效的 MET、AXL/MER 和 FGFR1/2/3 抑制剂,IC50 值低于 20 nM。
  47. GC19279 PD-166866 A potent inhibitor of FGFR1
  48. GC19187 H3B-6527 An FGFR4 inhibitor
  49. GC19156 TAS-120 An orally bioavailable, irreversible inhibitor of FGFRs
  50. GC19155 FGFR4-IN-1 An inhibitor of FGFR4
  51. GC19154 Roblitinib An FGFR4 inhibitor

Items 1 to 50 of 83 total

per page
  1. 1
  2. 2

Set Descending Direction