Dopamine Receptor(多巴胺受体)
Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.
Products for Dopamine Receptor
- Cat.No. 产品名称 Information
- GC14311 4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride dopamine release inhibitor
- GC16916 7-Hydroxy-PIPAT maleate D3 receptor agonist
- GC16574 7-Hydroxy-DPAT hydrobromide A dopamine D3 receptor agonist
- GC11945 BTCP maleate dopamine reuptake inhibitor
-
GC15856
3'-Fluorobenzylspiperone maleate
ligand for the D2 receptor
- GC13156 (+)-AJ 76 hydrochloride Dopamine receptor antagonist
- GC16049 AMI-193 AMI-193 (AMI-193) 是一种有效的、选择性的 5-HT2 和多巴胺 D2 受体拮抗剂,Kis 分别为 2 nM 和 3 nM。
- GC12456 GBR 12783 dihydrochloride GBR 12783 dihydrochloride 是一种特异性、有效和选择性的多巴胺摄取抑制剂,抑制大鼠和小鼠纹状体突触体对 [3H] 多巴胺的摄取,IC50 分别为 1.8 nM 和 1.2 nM。
- GC12179 GBR 13069 dihydrochloride dopamine uptake inhibitor
- GC14865 RuBi-Dopa dopamine receptor activator
- GC15326 Flupenthixol dihydrochloride Flupentixol 是一种具有口服活性的 D1/D2 多巴胺受体拮抗剂和新型 PI3K 抑制剂(PI3Kα;IC50=127 nM)。
- GC17075 NPEC-caged-dopamine Dopamine receptor agonist
- GC16267 6-Hydroxydopamine hydrobromide A catecholaminergic neurotoxin
- GC13573 Nomifensine An inhibitor of norepinephrine and dopamine reuptake
- GC17890 LE 300 A dopamine D1-like and 5-HT2A receptor antagonist
- GC17192 Quinelorane hydrochloride Quinelorane hydrochloride (LY163502) 是一种有效的多巴胺 D3/D2 受体激动剂。
- GC14048 SKF 38393 hydrobromide A partial agonist of dopamine D1-like receptors
- GC10349 (RS)-(±)-Sulpiride An atypical antipsychotic
- GC13931 Bromocriptine mesylate A dopamine receptor agonist
- GC13853 GBR 12935 dihydrochloride An inhibitor of dopamine uptake
- GC14657 Rotundine An antinociceptive alkaloid
- GC10441 Cabergoline A potent and selective dopamine D2 receptor agonist
- GC11028 Dopamine HCl An endogenous catecholamine
- GC10144 Domperidone A dopamine D2 receptor antagonist
- GC15107 Clomipramine HCl A tricyclic antidepressant
-
GC14216
Chlorpromazine HCl
A typical antipsychotic
- GC15546 Alizapride HCl A dopamine D2 receptor antagonist
- GC14759 Fenoldopam An agonist of dopamine D1A and D1B receptors
- GC15470 Levosulpiride 左舒必利 (RV-12309) 是舒必利的 (S)-对映异构体,是一种 D2 受体拮抗剂,是苯甲酰胺类的非典型抗精神病药物。
- GC16783 Pramipexole 2HCl Monohydrate Pramipexole 2HCl Monohydrate 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM .
- GC11960 Pramipexole Pramipexole 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM。
- GC10105 Amantadine HCl An NMDA receptor antagonist and antiviral agent
- GC15754 WAY-100635 Maleate A serotonin 5-HT1A antagonist
- GC13031 Trifluoperazine 2HCl An anti-adrenergic and anti-dopaminergic agent
- GC11462 Ropinirole HCl A dopamine D2 receptor agonist
- GC16615 Pergolide mesylate A dopamine D1 and D2 receptor agonist
- GC17600 PD128907 HCl A potent D3 receptor agonist
- GC10808 Droperidol A dopamine D2 and D4 receptor antagonist
- GC16229 Azaperone An Analytical Reference Standard
- GC17593 Lurasidone HCl An atypical antipsychotic
- GC16891 Quetiapine Fumarate An antagonist of diverse neurological receptors
- GC11182 LY404039 An agonist of mGluR2 and mGluR3
- GC10799 Iloperidone hydrochloride An atypical antipsychotic
- GC11186 Brexpiprazole A serotonin and dopamine receptor modulator
- GC10117 Aripiprazole An atypical antipsychotic
- GC12610 Amisulpride A dopamine D2 and D3 and 5-HT2B, 5-HT7, and 5-HT7A receptor antagonist
- GC12495 Olanzapine An atypical antipsychotic
- GC17760 Clozapine An atypical antipsychotic
- GC11506 Haloperidol hydrochloride A typical antipsychotic and dopamine D2-like receptor antagonist
- GC17599 Haloperidol A typical antipsychotic and dopamine D2-like receptor antagonist