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Dopamine Receptor(多巴胺受体)

Dopamine receptors (DR) are members of G protein-coupled receptors superfamily. There are 5 subtypes (D1, D2, D3, D4, D5) of DR which mediate the functions of dopamine in central nervous system for control of locomotion, cognition, and emotion etc.

Products for  Dopamine Receptor

  1. Cat.No. 产品名称 Information
  2. GC14311 4-Phenyl-1,2,3,4-tetrahydroisoquinoline hydrochloride dopamine release inhibitor
  3. GC16916 7-Hydroxy-PIPAT maleate D3 receptor agonist
  4. GC16574 7-Hydroxy-DPAT hydrobromide A dopamine D3 receptor agonist
  5. GC11945 BTCP maleate dopamine reuptake inhibitor
  6. GC15856 3'-Fluorobenzylspiperone maleate

    ligand for the D2 receptor

  7. GC13156 (+)-AJ 76 hydrochloride Dopamine receptor antagonist
  8. GC16049 AMI-193 AMI-193 (AMI-193) 是一种有效的、选择性的 5-HT2 和多巴胺 D2 受体拮抗剂,Kis 分别为 2 nM 和 3 nM。
  9. GC12456 GBR 12783 dihydrochloride GBR 12783 dihydrochloride 是一种特异性、有效和选择性的多巴胺摄取抑制剂,抑制大鼠和小鼠纹状体突触体对 [3H] 多巴胺的摄取,IC50 分别为 1.8 nM 和 1.2 nM。
  10. GC12179 GBR 13069 dihydrochloride dopamine uptake inhibitor
  11. GC14865 RuBi-Dopa dopamine receptor activator
  12. GC15326 Flupenthixol dihydrochloride Flupentixol 是一种具有口服活性的 D1/D2 多巴胺受体拮抗剂和新型 PI3K 抑制剂(PI3Kα;IC50=127 nM)。
  13. GC17075 NPEC-caged-dopamine Dopamine receptor agonist
  14. GC16267 6-Hydroxydopamine hydrobromide A catecholaminergic neurotoxin
  15. GC13573 Nomifensine An inhibitor of norepinephrine and dopamine reuptake
  16. GC17890 LE 300 A dopamine D1-like and 5-HT2A receptor antagonist
  17. GC17192 Quinelorane hydrochloride Quinelorane hydrochloride (LY163502) 是一种有效的多巴胺 D3/D2 受体激动剂。
  18. GC14048 SKF 38393 hydrobromide A partial agonist of dopamine D1-like receptors
  19. GC10349 (RS)-(±)-Sulpiride An atypical antipsychotic
  20. GC13931 Bromocriptine mesylate A dopamine receptor agonist
  21. GC13853 GBR 12935 dihydrochloride An inhibitor of dopamine uptake
  22. GC14657 Rotundine An antinociceptive alkaloid
  23. GC10441 Cabergoline A potent and selective dopamine D2 receptor agonist
  24. GC11028 Dopamine HCl An endogenous catecholamine
  25. GC10144 Domperidone A dopamine D2 receptor antagonist
  26. GC15107 Clomipramine HCl A tricyclic antidepressant
  27. GC14216 Chlorpromazine HCl

    A typical antipsychotic

  28. GC15546 Alizapride HCl A dopamine D2 receptor antagonist
  29. GC14759 Fenoldopam An agonist of dopamine D1A and D1B receptors
  30. GC15470 Levosulpiride 左舒必利 (RV-12309) 是舒必利的 (S)-对映异构体,是一种 D2 受体拮抗剂,是苯甲酰胺类的非典型抗精神病药物。
  31. GC16783 Pramipexole 2HCl Monohydrate Pramipexole 2HCl Monohydrate 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM .
  32. GC11960 Pramipexole Pramipexole 是一种选择性和血脑屏障 (BBB) 渗透性多巴胺 D2 型受体激动剂,对 D2 型受体、D2、D3 和 D4 受体的 Kis 分别为 2.2 nM、3.9 nM、0.5 nM 和 1.3 nM。
  33. GC10105 Amantadine HCl An NMDA receptor antagonist and antiviral agent
  34. GC15754 WAY-100635 Maleate A serotonin 5-HT1A antagonist
  35. GC13031 Trifluoperazine 2HCl An anti-adrenergic and anti-dopaminergic agent
  36. GC11462 Ropinirole HCl A dopamine D2 receptor agonist
  37. GC16615 Pergolide mesylate A dopamine D1 and D2 receptor agonist
  38. GC17600 PD128907 HCl A potent D3 receptor agonist
  39. GC10808 Droperidol A dopamine D2 and D4 receptor antagonist
  40. GC16229 Azaperone An Analytical Reference Standard
  41. GC17593 Lurasidone HCl An atypical antipsychotic
  42. GC16891 Quetiapine Fumarate An antagonist of diverse neurological receptors
  43. GC11182 LY404039 An agonist of mGluR2 and mGluR3
  44. GC10799 Iloperidone hydrochloride An atypical antipsychotic
  45. GC11186 Brexpiprazole A serotonin and dopamine receptor modulator
  46. GC10117 Aripiprazole An atypical antipsychotic
  47. GC12610 Amisulpride A dopamine D2 and D3 and 5-HT2B, 5-HT7, and 5-HT7A receptor antagonist
  48. GC12495 Olanzapine An atypical antipsychotic
  49. GC17760 Clozapine An atypical antipsychotic
  50. GC11506 Haloperidol hydrochloride A typical antipsychotic and dopamine D2-like receptor antagonist
  51. GC17599 Haloperidol A typical antipsychotic and dopamine D2-like receptor antagonist

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