PAR1
PAR1 (protease-activated receptor 1) is a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain.
- Cat.No. 产品名称 Information
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GC65529
TRAP-6 amide
A peptide PAR1 agonist
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GC65439
GB-88
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GC65312
AZ8838
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GC64979
I-191
I-191 is a potent PAR2 antagonist that inhibits multiple PAR2-induced signaling pathways and functional responses. I-191 also inhibits ERK1/2 phosphorylation, RhoA activation, and inhibition of forskolin-stimulated cAMP accumulation induced by micromolar concentrations of biased ligand GB88.
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GC64347
Vorapaxar sulfate
A PAR1 antagonist
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GC63658
Atopaxar
Atopaxar(E5555,ER-172594-00) is a potent, orally active, selective and reversible thrombin receptor protease-activated receptor-1 (PAR-1) antagonist.
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GC63540
SCH79797
An antagonist of PAR1
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GC62469
Protease-Activated Receptor-1, PAR-1 Agonist TFA
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GC62101
PAR-2-IN-1
IUN76750 is a PAR-2 signaling pathway inhibitor.
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GC61777
RWJ-56110 dihydrochloride
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GC61501
FSLLRY-NH2 TFA
FSLLRY-NH2 TFA (FSY-NH2) is a selective protease-activated receptor 2 (PAR2) inhibitor with an ic50 of 50 ?M in PAR2-KNRK cells.
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GC61456
Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA
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GC61316
tcY-NH2 TFA
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GC60807
ENMD-1068 hydrochloride
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GC38731
2-Furoyl-LIGRLO-amide TFA
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GC38329
GB-110 hydrochloride
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GA23350
PAR-3 (1-6) amide (human)
A peptide agonist of PAR1 and PAR2
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GC37852
UDM-001651
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GC37770
TFLLR-NH2(TFA)
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GC36125
GB-110
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GC33599
PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA))
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GC33429
Protease-Activated Receptor-4
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GC18717
BMS 986120
A selective PAR4 antagonist
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GC18152
AZ-3451
A PAR2 antagonist
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GC10291
SCH 79797 dihydrochloride
An antagonist of PAR1
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GC17545
Vorapaxar
A PAR1 antagonist
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GC14540
SLIGKV-NH2
SLIGKV-NH2 (SLIGKV-NH2) 是一种高效的蛋白酶激活受体 2 (PAR2) 激活肽。
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GC17368
2-Furoyl-LIGRLO-amide
A potent agonist of PAR2
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GC11662
TRAP-6
TRAP-6 (PAR-1 agonist peptide) 是一种肽片段,是一种选择性蛋白酶激活受体 1 (PAR1) 激动剂。
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GC11951
PAR 4 (1-6)
A peptide agonist of PAR4
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GC13227
LRGILS-NH2
LRGILS-NH2 是一种反向序列蛋白酶激活受体-2 (PAR-2)-失活的阴性对照,SLIGRL-NH2 是一种 PAR-2 激活肽。
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GC17991
RLLFT-NH2
RLLFT-NH2 是 TFLLR-NH2 的反向氨基酸序列阴性对照肽。
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GC11727
VKGILS-NH2
VKGILS-NH2 是 SLIGKV-NH2(蛋白酶激活受体 2 (PAR2) 激动剂)的反向氨基酸序列控制肽。
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GC14831
AC 264613
An agonist of PAR2
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GC15290
AC 55541
A selective PAR2 agonist
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GC10140
Thrombin Receptor Agonist Peptide
A peptide agonist of the α-thrombin receptor
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GC15817
PAR-4 Agonist Peptide, amide (AY-NH2)
PAR-4 Agonist Peptide, amide(AY-NH2) (PAR-4-AP; AY-NH2) 是一种蛋白酶激活的受体 4 (PAR-4) 激动剂,对 PAR-1 或 PAR- 均无影响2 并且其作用被 PAR-4 拮抗剂阻断。
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GC17444
TFLLR-NH2
A peptide agonist of PAR1
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GC17514
SLIGRL-NH2
A PAR2 agonist
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GC13004
ML161
Reversible inhibitor of PAR1-mediated platelet activation
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GP10085
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
凝血酶受体激活剂 5 (TRAP-5) 也称为凝血因子 II 受体 (1-5) 或蛋白酶激活受体 1 (1-5),用于研究冠心病 (CHD)。