HIV(人类免疫缺陷病毒)
HIV (human immunodeficiency virus) is a lentivirus that infect immune system. It cause immune system failure and lead to AIDS (acquired immnudeficiency syndrome).
Products for HIV
- Cat.No. 产品名称 Information
- GC14454 Tipranavir A nonpeptidic HIV protease inhibitor
- GC15785 Saquinavir mesylate An HIV protease inhibitor
- GC15335 Saquinavir Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,用于抗逆转录病毒治疗。
- GC11059 Rilpivirine A non-nucleoside reverse transcriptase inhibitor
- GC14084 Nelfinavir Mesylate An HIV-1 protease inhibitor
- GC16035 NBD-556 A small molecule CD4 mimetic
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GC16589
Limonin
A limonoid
- GC16596 Lersivirine An NNRTI
- GC12998 HIV-1 integrase inhibitor HIV-1整合酶抑制剂可用于抗HIV。
- GC12555 GS-9620 A TLR7 agonist
- GC11300 Fosamprenavir Calcium Salt A prodrug form of amprenavir
- GC16063 Flavopiridol An inhibitor of cyclin-dependent kinases
- GC12871 CDK9 inhibitor CDK9 inhibitor 是一种新型的选择性 CDK9 抑制剂,用于治疗 HIV 感染,对 CDK9/CycT1 的 IC50 为 39 nM,从参考化合物 87 中提取。
- GC13119 BMS-663068 BMS-663068 (BMS-663068) 是 BMS-626529 的膦酰氧基甲基前药。
- GC10794 BMS-626529 An HIV-1 attachment inhibitor
- GC10480 Betulinic acid A plant triterpenoid similar to bile acids
- GC12196 AMD-070 A CXCR4 antagonist
- GC13805 Abacavir 阿巴卡韦是一种具有口服活性和竞争性的核苷类逆转录酶抑制剂。
- GC16629 Rolipram A phosphodiesterase-4 inhibitor
- GC14269 Cobicistat (GS-9350) An inhibitor of CYP3A
- GC12426 Birinapant (TL32711) An antagonist of cIAP1, cIAP2, and XIAP
- GC15050 Deuterated Atazanivir-D3-3 HIV-1 protease inhibitor
- GC11772 Deuterated Atazanivir-D3-2 HIV-1 protease inhibitor
- GC15984 Deuterated Atazanivir-D3-1 HIV-1 protease inhibitor
- GC14152 Amprenavir (agenerase) A selective HIV protease inhibitor
- GC16602 Darunavir An HIV-1 protease inhibitor
- GC17303 Ritonavir An HIV protease inhibitor
- GC10240 Atazanavir sulfate (BMS-232632-05) An inhibitor of HIV-1 protease
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GC12945
Atazanavir
An inhibitor of HIV-1 protease
- GC15794 Valproic acid sodium salt (Sodium valproate) A class I HDAC inhibitor
- GC17906 S/GSK1349572 A potent inhibitor of HIV integrase
- GC11956 Raltegravir (MK-0518) Raltegravir (MK-0518) 是一种有效的整合酶 (IN) 抑制剂,用于治疗 HIV 感染。
- GC15561 MK-2048 MK-2048 是一种有效的整合酶和 INR263K 抑制剂,IC50 分别为 2.6 nM 和 1.5 nM。
- GC14466 Fluorouracil (Adrucil) A prodrug form of FdUMP
- GC14996 Elvitegravir (GS-9137) An inhibitor of HIV-1 integrase
- GC11923 BMS-707035 BMS-707035 是一种有效的口服活性 HIV-1 整合酶链转移抑制剂 (INSTI)。
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GC17390
Vorinostat (SAHA, MK0683)
An HDAC inhibitor
- GN10113 Cepharanthine A biscoclaurine alkaloid
- GN10216 Shikonin A natural product with anti-inflammatory and anti-tumor activity
- GN10184 Oleanolic acid A pentacyclic triterpenoid with diverse biological activities
- GN10018 Baicalin A flavonoid with diverse biological activities
- GN10001 Sennoside A A dianthrone glycoside with laxative and gastroprotective activities
- GN10451 Psoralen A photoactive probe to study DNA
- GC12257 Panobinostat (LBH589) A pan-HDAC inhibitor
- GC13716 Lopinavir A potent HIV-1 protease inhibitor
- GC14049 (-)-Epigallocatechin gallate (EGCG) (-)-Epigallocatechin Gallate sulfate (EGCG) 是绿茶中的一种主要多酚,可抑制细胞增殖并诱导细胞凋亡。此外,它还能抑制谷氨酸脱氢酶1/2 (GDH1/2, GLUD1/2)的活性。.