FAK(局部粘着斑激酶)
FAK (focal adhesion kinase), also known as PTK2, is a focal adhesion-associated protein kinase involved in cellular adhesion and spreading processes.
- Cat.No. 产品名称 Information
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GC68463
ULK1-IN-2
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GC68030
FAK-IN-7
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GC65886
BI-853520
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GC65457
BI-3663
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GC64992
YH-306
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GC64888
GSK215
GSK215 is a potent and selective PROTAC focal adhesion kinase (FAK) degrader, which exerts FAK degradation in A549 non-small-cell lung cancer cells with DC50 of 1.3 nM by a strong time-dependence way and maximal degradation (Dmax) near the limit of the assay quantification (Dmax 99%).
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GC64377
Batatasin III
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GC64015
AMP-945
AMP-945 is an inhibitor of the focal adhesion kinase (FAK).
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GC62111
PND-1186 hydrochloride
A potent FAK inhibitor
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GC38437
Fangchinoline
An alkaloid with diverse biological activities
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GC36985
PROTAC FAK degrader 1
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GC36025
FAK inhibitor 2
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GC35827
Defactinib hydrochloride
A FAK inhibitor
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GC35728
Conteltinib
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GC44605
Petunidin (chloride)
An O-methylated anthocyanidin
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GC34488
BI-4464
BI-4464 is a highly selective ATP competitive inhibitor of PTK2/FAK, with an IC50 of 17 nM.
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GC33045
NAMI-A
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GC32979
Chloropyramine hydrochloride
Chloropyramine hydrochloride (Halopyramine) is a histamine receptor H1 antagonist and has anti-cholinergic, antispasmodic, and antiallergic effects.
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GC19179
GSK2256098
A FAK inhibitor
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GC17500
SU6656
Inhibitor of Src kinases
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GC16813
Defactinib
A FAK inhibitor
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GC14489
Y 11
An inhibitor of FAK1
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GC12174
FAK Inhibitor 14
An inhibitor of the FAK1
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GC11107
PF-573228
A selective focal adhesion kinase inhibitor
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GC15273
CEP-37440
A dual inhibitor of FAK1 and ALK
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GC14407
PF-431396
A FAK/PYK2 dual inhibitor
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GC16821
TAE226(NVP-TAE226)
A dual inhibitor of FAK and IGF-1R
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GC10810
PF-562271 HCl
PF-562271 (VS-6062) hydrochloride 是一种有效的 ATP 竞争性和可逆的 FAK 和 Pyk2 激酶抑制剂,IC50 分别为 1.5 nM 和 13 nM。
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GC14767
PF-00562271
A selective FAK/PYK2 inhibitor
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GC15380
PF-562271
A selective FAK/PYK2 inhibitor
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GC13410
Masitinib (AB1010)
An inhibitor of c-Kit
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GC15164
PND-1186
A potent FAK inhibitor