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Raf

Raf is a family of three serine/threonine-specific protein kinases that are related to retroviral oncogenes.

Products for  Raf

  1. Cat.No. 产品名称 Information
  2. GC10505 GDC-0879 An inhibitor of B-RafV600E
  3. GC16499 Sorafenib Tosylate A multi-kinase inhibitor
  4. GC10111 Regorafenib A multi-kinase inhibitor
  5. GC17455 TAK-632 A selective pan-Raf inhibitor
  6. GC14534 Regorafenib monohydrate A multi-kinase inhibitor
  7. GC14606 Regorafenib hydrochloride A multi-kinase inhibitor
  8. GC11649 MLN 2480 An oral pan-Raf kinase inhibitor
  9. GC12486 Dabrafenib Mesylate (GSK-2118436) A Raf kinase inhibitor
  10. GC17860 CEP-32496 hydrochloride A potent inhibitor of B-Raf
  11. GC12151 B-Raf inhibitor B-Raf inhibitor 是一种有效的双重 TGFβ-activated kinase 1 (TAK1) 和 mitogen-activated protein kinase kinase kinase 2 (MAP4K2) 抑制剂,IC50 分别为 41.1 nM 和 18.2 nM。
  12. GC12482 BRAF inhibitor BRAF 抑制剂是从专利 WO/2011103196 A1 化合物 P-0850 中提取的 B-Raf 抑制剂。
  13. GC14732 PLX-4720 An orally-available inhibitor of the B-raf mutant B-RafV600E
  14. GC17369 Sorafenib

    Sorafenib acts as a multi-kinase inhibitor, targeting Raf-1 and B-Raf with IC50 values of 6 nM and 22 nM, respectively.

  15. GC13412 Vemurafenib (PLX4032, RG7204)

    An inhibitor of mutant V600E and wild type B-Raf

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