Raf
Raf is a family of three serine/threonine-specific protein kinases that are related to retroviral oncogenes.
Products for Raf
- Cat.No. 产品名称 Information
- GC10505 GDC-0879 An inhibitor of B-RafV600E
- GC16499 Sorafenib Tosylate A multi-kinase inhibitor
- GC10111 Regorafenib A multi-kinase inhibitor
- GC17455 TAK-632 A selective pan-Raf inhibitor
- GC14534 Regorafenib monohydrate A multi-kinase inhibitor
- GC14606 Regorafenib hydrochloride A multi-kinase inhibitor
- GC11649 MLN 2480 An oral pan-Raf kinase inhibitor
- GC12486 Dabrafenib Mesylate (GSK-2118436) A Raf kinase inhibitor
- GC17860 CEP-32496 hydrochloride A potent inhibitor of B-Raf
- GC12151 B-Raf inhibitor B-Raf inhibitor 是一种有效的双重 TGFβ-activated kinase 1 (TAK1) 和 mitogen-activated protein kinase kinase kinase 2 (MAP4K2) 抑制剂,IC50 分别为 41.1 nM 和 18.2 nM。
- GC12482 BRAF inhibitor BRAF 抑制剂是从专利 WO/2011103196 A1 化合物 P-0850 中提取的 B-Raf 抑制剂。
- GC14732 PLX-4720 An orally-available inhibitor of the B-raf mutant B-RafV600E
-
GC17369
Sorafenib
Sorafenib acts as a multi-kinase inhibitor, targeting Raf-1 and B-Raf with IC50 values of 6 nM and 22 nM, respectively.
-
GC13412
Vemurafenib (PLX4032, RG7204)
An inhibitor of mutant V600E and wild type B-Raf