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5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC14392 SB 242084 Specific antagonist of 5-HT2C
  3. GC11384 BTS 54-505 hydrochloride Potent SNRI,sibutramine metabolite
  4. GC11176 2-Methyl-5-hydroxytryptamine hydrochloride 2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。
  5. GC17826 Tegaserod maleate A potent 5-HT4 agonist
  6. GC15367 EMDT oxalate EMDT 草酸盐是一种选择性 5-HT6 激动剂,具有抗抑郁作用。
  7. GC10051 MDL 100907 Selective antagonist of the serotonin receptor 5-HT2A
  8. GC15660 SB 399885 hydrochloride A 5-HT6 receptor antagonist
  9. GC16324 Nefazodone hydrochloride A serotonin, norepinephrine, and dopamine reuptake inhibitor
  10. GC13109 Fananserin Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂,对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。
  11. GC11495 Lofepramine A tricyclic antidepressant
  12. GC14583 R 59-022 A DGK inhibitor
  13. GC16735 (±)-McN 5652

    5-HT uptake inhibitor

  14. GC18102 Paroxetine maleate 5-HT uptake inhibitor
  15. GC17525 AS 19

    A 5-HT7 receptor agonist

  16. GC13883 Ritanserin A potent 5-HT2A receptor antagonist
  17. GC13133 Ipsapirone A partial agonist of serotonin 5-HT1A receptors
  18. GC18013 S 14506 hydrochloride A 5-HT1A receptor agonist
  19. GC10630 Zimelidine dihydrochloride

    5-HT re-uptake inhibitor

  20. GC14093 Indatraline hydrochloride Indatraline hydrochloride (Lu 19-005) 是一种非选择性单胺转运蛋白抑制剂,可阻断神经递质(多巴胺、血清素和去甲肾上腺素)的再摄取,其功效与可卡因相似。
  21. GC14035 Citalopram hydrobromide A selective serotonin reuptake inhibitor
  22. GC11624 GR 113808 A 5-HT4 antagonist
  23. GC14805 (S)-WAY 100135 dihydrochloride A 5-HT1A receptor antagonist
  24. GC13438 SB 224289 hydrochloride A 5-HT1B receptor inverse agonist
  25. GC17333 (R)-(+)-8-Hydroxy-DPAT hydrobromide 5-HT1A serotonin receptor agonist
  26. GC12632 Cyanopindolol hemifumarate 5-HT1A/1B antagonist and β-adrenoceptor antagonist
  27. GC11984 Isamoltane hemifumarate Isamoltane hemifumarate 是 5-HT1B 受体的选择性拮抗剂,抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B 识别位点的结合,IC50 为 39 nM。
  28. GC14891 MM 77 dihydrochloride MM 77 dihydrochloride 是一种有效的 5-HT1A 受体的突触后拮抗剂。
  29. GC17477 5-Nonyloxytryptamine oxalate A potent 5-HT1Dβ receptor agonist
  30. GC12427 8-Hydroxy-PIPAT oxalate 5-HT1A receptor agonist
  31. GC14008 Anpirtoline hydrochloride 5-HT1B receptor agonist
  32. GC12276 CGS 12066B dimaleate A 5-HT1B receptor agonist
  33. GC10357 Metergoline A serotonin receptor antagonist
  34. GC15311 BP 554 maleate Selective 5-HT1A agonist
  35. GC15235 NAN-190 hydrobromide A 5-HT1A receptor mixed antagonist and partial agonist
  36. GC14966 8-Hydroxy-DPAT hydrobromide A 5-HT1A receptor agonist
  37. GC16135 Cinanserin hydrochloride A 5-HT receptor antagonist
  38. GC10985 MDL 72832 hydrochloride ligand for 5-HT1A receptor, potent and selective
  39. GC14019 MDL 73005EF hydrochloride 5-HT1A receptor antagonist
  40. GC14105 Alprenolol hydrochloride A non-selective β-AR and 5-HT receptor antagonist
  41. GC17854 PNU 142633 PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂,对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
  42. GC17734 Pindolol A β1- and β2-AR antagonist
  43. GC14083 MDL 72222 MDL 72222 (MDL 72222) 是一种选择性 5-HT3 受体拮抗剂,IC50 为 0.33 nM。
  44. GC14657 Rotundine An antinociceptive alkaloid
  45. GC15639 Ramosetron Hydrochloride A potent, selective 5-HT3 receptor antagonist
  46. GC16202 Sarpogrelate hydrochloride A selective 5-HT2 receptor antagonist
  47. GC14558 Dihydroergotamine mesylate An agonist of 5-HT1B and 5-HT1D receptors
  48. GC14563 Ketanserin A potent 5-HT2 receptor antagonist
  49. GC11191 Buspirone HCl An Analytical Reference Standard
  50. GC17974 Latrepirdine dihydrochloride A neuroprotective agent
  51. GC17061 Dapoxetine HCl An Analytical Reference Standard

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