5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
Products for 5-HT Receptor
- Cat.No. 产品名称 Information
- GC14392 SB 242084 Specific antagonist of 5-HT2C
- GC11384 BTS 54-505 hydrochloride Potent SNRI,sibutramine metabolite
- GC11176 2-Methyl-5-hydroxytryptamine hydrochloride 2-Methyl-5-hydroxytryptamine hydrochloride (2-Methyl-5-hydroxytryptamine hydrochloride) 是一种有效的选择性 5-HT3 受体激动剂。
- GC17826 Tegaserod maleate A potent 5-HT4 agonist
- GC15367 EMDT oxalate EMDT 草酸盐是一种选择性 5-HT6 激动剂,具有抗抑郁作用。
- GC10051 MDL 100907 Selective antagonist of the serotonin receptor 5-HT2A
- GC15660 SB 399885 hydrochloride A 5-HT6 receptor antagonist
- GC16324 Nefazodone hydrochloride A serotonin, norepinephrine, and dopamine reuptake inhibitor
- GC13109 Fananserin Fananserin (RP 62203) 是一种口服有效的选择性 5-hydroxytryptamine2 (5-HT2) 受体拮抗剂,对大鼠 5-HT2A 受体的 Ki 值为 0.37 nM。
- GC11495 Lofepramine A tricyclic antidepressant
- GC14583 R 59-022 A DGK inhibitor
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GC16735
(±)-McN 5652
5-HT uptake inhibitor
- GC18102 Paroxetine maleate 5-HT uptake inhibitor
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GC17525
AS 19
A 5-HT7 receptor agonist
- GC13883 Ritanserin A potent 5-HT2A receptor antagonist
- GC13133 Ipsapirone A partial agonist of serotonin 5-HT1A receptors
- GC18013 S 14506 hydrochloride A 5-HT1A receptor agonist
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GC10630
Zimelidine dihydrochloride
5-HT re-uptake inhibitor
- GC14093 Indatraline hydrochloride Indatraline hydrochloride (Lu 19-005) 是一种非选择性单胺转运蛋白抑制剂,可阻断神经递质(多巴胺、血清素和去甲肾上腺素)的再摄取,其功效与可卡因相似。
- GC14035 Citalopram hydrobromide A selective serotonin reuptake inhibitor
- GC11624 GR 113808 A 5-HT4 antagonist
- GC14805 (S)-WAY 100135 dihydrochloride A 5-HT1A receptor antagonist
- GC13438 SB 224289 hydrochloride A 5-HT1B receptor inverse agonist
- GC17333 (R)-(+)-8-Hydroxy-DPAT hydrobromide 5-HT1A serotonin receptor agonist
- GC12632 Cyanopindolol hemifumarate 5-HT1A/1B antagonist and β-adrenoceptor antagonist
- GC11984 Isamoltane hemifumarate Isamoltane hemifumarate 是 5-HT1B 受体的选择性拮抗剂,抑制 [125I]ICYP 与大鼠脑膜中 5-HT1B 识别位点的结合,IC50 为 39 nM。
- GC14891 MM 77 dihydrochloride MM 77 dihydrochloride 是一种有效的 5-HT1A 受体的突触后拮抗剂。
- GC17477 5-Nonyloxytryptamine oxalate A potent 5-HT1Dβ receptor agonist
- GC12427 8-Hydroxy-PIPAT oxalate 5-HT1A receptor agonist
- GC14008 Anpirtoline hydrochloride 5-HT1B receptor agonist
- GC12276 CGS 12066B dimaleate A 5-HT1B receptor agonist
- GC10357 Metergoline A serotonin receptor antagonist
- GC15311 BP 554 maleate Selective 5-HT1A agonist
- GC15235 NAN-190 hydrobromide A 5-HT1A receptor mixed antagonist and partial agonist
- GC14966 8-Hydroxy-DPAT hydrobromide A 5-HT1A receptor agonist
- GC16135 Cinanserin hydrochloride A 5-HT receptor antagonist
- GC10985 MDL 72832 hydrochloride ligand for 5-HT1A receptor, potent and selective
- GC14019 MDL 73005EF hydrochloride 5-HT1A receptor antagonist
- GC14105 Alprenolol hydrochloride A non-selective β-AR and 5-HT receptor antagonist
- GC17854 PNU 142633 PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂,对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
- GC17734 Pindolol A β1- and β2-AR antagonist
- GC14083 MDL 72222 MDL 72222 (MDL 72222) 是一种选择性 5-HT3 受体拮抗剂,IC50 为 0.33 nM。
- GC14657 Rotundine An antinociceptive alkaloid
- GC15639 Ramosetron Hydrochloride A potent, selective 5-HT3 receptor antagonist
- GC16202 Sarpogrelate hydrochloride A selective 5-HT2 receptor antagonist
- GC14558 Dihydroergotamine mesylate An agonist of 5-HT1B and 5-HT1D receptors
- GC14563 Ketanserin A potent 5-HT2 receptor antagonist
- GC11191 Buspirone HCl An Analytical Reference Standard
- GC17974 Latrepirdine dihydrochloride A neuroprotective agent
- GC17061 Dapoxetine HCl An Analytical Reference Standard