HER2
HER2 is a member of the epidermal growth factor. It initiates the EGF downstream cascade by forming a heterodimer with other ligand-bound EGF receptor. It is associated with breast and ovarian cancers.
- Cat.No. 产品名称 Information
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GC13257
AC480 (BMS-599626)
A dual inhibitor of EGFR and HER2
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GC10707
Afatinib dimaleate
An inhibitor of EGFR and ErbB2
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GC13296
Afatinib(BIBW2992)
A selective dual inhibitor of EGFR/HER2
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GC10606
BMS-599626 Hydrochloride
BMS-599626 Hydrochloride (AC480 Hydrochloride) 是一种选择性的口服生物可利用的 HER1 和 HER2 抑制剂,IC50 分别为 20 和 30 nM。 BMS-599626 Hydrochloride 对 HER4 (IC50=190 nM) 的效力降低约 8 倍,对 VEGFR2、c-Kit、Lck、MEK 的效力超过 100 倍。 BMS-599626 Hydrochloride 抑制肿瘤细胞增殖,并有可能增加肿瘤对放疗的反应。
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GC12087
Canertinib dihydrochloride
A pan-ErbB tyrosine kinase inhibitor
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GC13091
CP-724714
A selective HER2/ErbB2 tyrosine kinase inhibitor
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GC16008
CUDC-101
A multi-target inhibitor of HDACs, EGFR, and HER2
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GC13608
Lapatinib
A dual inhibitor of EGFR and ErbB2
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GC16593
Lapatinib Ditosylate
Lapatinib Ditosylate (GW572016 ditosylate monohydrate) 是有效的 ErbB-2 和 EGFR 酪氨酸激酶结构域抑制剂,对纯化的 EGFR 和 ErbB-2 的 IC50 值分别为 10.2 和 9.8 nM。
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GC10250
Mubritinib (TAK 165)
A selective inhibitor of HER2
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GC10362
Neratinib (HKI-272)
A dual inhibitor of EGFR and HER2
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GC17473
Pelitinib (EKB-569)
An EGFR receptor tyrosine kinase inhibitor
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GC17916
Poziotinib
An inhibitor of EGFRs
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GC11172
TAK-285
A dual inhibitor of EGFR and HER2
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GC15271
Tyrphostin AG 879
A non-specific tyrphostin ErbB2 inhibitor