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BMX Kinase(BMX激酶)

Bmx kinase is a member of Tec kinase family. It is involved in different signaling pathways and controls differential and tumorigenicity in several cancer types.

  1. Cat.No. 产品名称 Information
  2. GC35684 CHMFL-EGFR-202 CHMFL-EGFR-202 是一种有效、不可逆的表皮生长因子受体 (EGFR) 突变型激酶抑制剂, 对 耐药突变型 EGFR T790M 和 WT EGFR 激酶作用的 IC50 值分别为 5.3 nM 和 8.3 nM。在细胞中,CHMFL-EGFR-202 对 EGFR L858R/T790M 的选择性是 EGFR 野生型的 10 倍。CHMFL-EGFR-202 以 “DFG-in-C-helix-out” 的不活跃结合构象形式共价结合 EGFR,对 EGFR 突变体驱动的非小细胞肺癌 (NSCLC) 细胞株具有较强的抗增殖作用。
  3. GC33020 CHMFL-BMX-078 (CHMFL-BMX 078) An irreversible BMX inhibitor
  4. GC11063 BMX-IN-1 A selective BMX and BTK inhibitor

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