EZH2(zeste 同源物 2增强子)

EZH2 (enhancer of zeste homolog 2) is a polycomb group protein and histone methyltrasferase that associated with transcriptional repression. It catalyzes trimethylation of H3K27me3 (histone H3 lysine 27) as a catalytic subunit of PRC2 (polycomb repressive complex 2).

Cat.No. 产品名称 Information
GC11414 GSK503 A potent, selective EZH2 inhibitor
GC11484 CPI-169 S-enantiomer EZH2 inhibitor
GC12146 CPI-169 R-enantiomer EZH2 inhibitor
GC16599 CPI-169 A selective EZH2 inhibitor
GC14756 EI1 A selective inhibitor of EZH2
GC17534 GSK343 A selective, cell-permeable EZH2 inhibitor
GC15783 GSK126
A selective EZH2 inhibitor
GC13878 EPZ005687 A potent, selective inhibitor of EZH2
GC17907 3-Deazaneplanocin A (DZNep) hydrochloride An inhibitor of the lysine methyltransferase EZH2
GC13145 3-Deazaneplanocin,DZNep
An inhibitor of lysine methyltransferase EZH2