MELK(母体胚胎亮氨酸拉链激酶)
MELK (maternal embryonic leucine zipper kinase) is an enzyme that interacts with CDC25B.
- Cat.No. 产品名称 Information
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GC69242
HTH-01-091
HTH-01-091 是一种强效且选择性的 maternal embryonic leucine zipper kinase (MELK) 抑制剂,其 IC50 为 10.5 nM。HTH-01-091 还能抑制 PIM1/2/3、RIPK2、DYRK3、smMLCK 和 CLK2。HTH-01-091 可用于乳腺癌研究。
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GC25626
MELK-8a Dihydrochloride
MELK-8a Dihydrochloride is a novel inhibitor of maternal embryonic leucine zipper kinase (MELK) with an IC50 of 2 nM.
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GC66065
MELK-IN-1
MELK-IN-1是母体胚胎亮氨酸拉链激酶 (MELK)的有效抑制剂,IC50 和 Ki 分别为3 nM和0.39 nM。
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GC32995
JNJ-47117096 hydrochloride (MELK-T1 hydrochloride)
JNJ-47117096 hydrochloride (MELK-T1 hydrochloride) 是有效的选择性 MELK 抑制剂,IC50 为 23 nM,也有效抑制 Flt3,IC50 为 18 nM。
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GC32736
MELK-8a hydrochloride
A MELK inhibitor
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GC12155
OTSSP167 hydrochloride
A potent inhibitor of MELK
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GC10201
OTSSP167
A potent inhibitor of MELK