MELK(母体胚胎亮氨酸拉链激酶)
MELK (maternal embryonic leucine zipper kinase) is an enzyme that interacts with CDC25B.
Products for MELK
- Cat.No. 产品名称 Information
- GC69242 HTH-01-091 HTH-01-091 是一种强效且选择性的 maternal embryonic leucine zipper kinase (MELK) 抑制剂,其 IC50 为 10.5 nM。HTH-01-091 还能抑制 PIM1/2/3、RIPK2、DYRK3、smMLCK 和 CLK2。HTH-01-091 可用于乳腺癌研究。
- GC25626 MELK-8a Dihydrochloride MELK-8a Dihydrochloride is a novel inhibitor of maternal embryonic leucine zipper kinase (MELK) with an IC50 of 2 nM.
- GC66065 MELK-IN-1 MELK-IN-1是母体胚胎亮氨酸拉链激酶 (MELK)的有效抑制剂,IC50 和 Ki 分别为3 nM和0.39 nM。
- GC32995 JNJ-47117096 hydrochloride (MELK-T1 hydrochloride) JNJ-47117096 hydrochloride (MELK-T1 hydrochloride) 是有效的选择性 MELK 抑制剂,IC50 为 23 nM,也有效抑制 Flt3,IC50 为 18 nM。
- GC32736 MELK-8a hydrochloride A MELK inhibitor
- GC12155 OTSSP167 hydrochloride A potent inhibitor of MELK
- GC10201 OTSSP167 A potent inhibitor of MELK