Adrenergic Receptor(肾上腺素能受体)
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Products for Adrenergic Receptor
- Cat.No. 产品名称 Information
- GC12188 Salmefamol β2-adrenergic receptor agonist
- GC30092 Salmeterol (GR33343X) Salmeterol (Astmerole, GR-33343X, SN408D) is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500).
- GC11531 Salmeterol xinafoate A long-acting β2-adrenergic receptor agonist
- GC48067 Salmeterol-d3 An internal standard for the quantification of salmeterol
- GC14220 Scopine A metabolite of scopolamine
- GC11373 Scopine HCl A metabolite of scopolamine
- GC13623 SDZ 21009 β-adrenoceptor and 5-HT1A/1B receptor antagonist
- GC13990 Setiptiline Setiptiline (Org-8282) 是一种血清素受体拮抗剂。
- GC13549 Setiptiline maleate Setiptiline maleate (MO-8282 maleate) 是一种血清素受体拮抗剂。
- GC15719 Silodosin A potent α1A-adrenoceptor antagonist
- GC12856 SKF 86466 hydrochloride An α2-AR antagonist
- GC15426 SNAP 5089 α1A-adrenoceptor antagonist
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GC34808
Solabegron
Solabegron(GW427353)是β3肾上腺素能受体(β3-AR)的选择性激动剂,在中国仓鼠卵巢细胞中测得的EC50值为22nM。目前正在被用于开发治疗膀胱过度活跃和肠易激综合征。
- GC13173 Sotalol An Analytical Reference Standard
- GC15631 Sotalol hydrochloride A β-AR antagonist and a class III antiarrhythmic agent
- GC45893 Sotalol-d6 (hydrochloride) An internal standard for the quantification of sotalol
- GC31005 Spirendolol (Li 32-468) Spirendolol (Li 32-468) is a ⋲肾上腺素受体拮抗剂。
- GC13338 Spiroxatrine 5-HT1A拮抗剂和α2C肾上腺素能受体拮抗剂
- GC16091 SR 58611A hydrochloride A selective β3-AR agonist
- GC12227 SR 59230A hydrochloride A β3-AR antagonist
- GC39725 SR59230A A β3-AR antagonist
- GC11913 ST 91 α2-adrenoceptor agonist
- GC38438 Synephrine Synephrine (Oxedrine), a natural protoalkaloid in the extract of bitter orange and other citrus species, is commonly used for weight loss.
- GC12715 Synephrine HCl An alkaloid
- GC39449 Tamsulosin A potent α1-AR antagonist
- GC50035 Tamsulosin hydrochloride A potent α1-AR antagonist
- GC65276 Tasipimidine sulfate Tasipimidine sulfate 是一种具有口服活性的、选择性的 α2A-adrenoceptor 激动剂,对人 α2A-adrenoceptor 的pEC50 为 7.57。Tasipimidine sulfate 可用于情境焦虑和恐惧的研究。
- GC16217 TC-G 1000 α2D-adrenoceptor agonist
- GC31453 TD-5471 hydrochloride TD-5471hydrochloride是一种有效的选择性人β2肾上腺素能受体的全激动剂。
- GC30273 Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) Tedatioxetine (Lu AA24530) hydrobromide 可作为 5-HT2A、5-HT2C、5-HT3 和 α;1A-肾上腺素受体拮抗剂,可作为 5-羟色胺和去甲肾上腺素 (NE) 的首选三重再摄取抑制剂 (TRI)。
- GC30458 Teoprolol Teoprolol是一种β-adrenergic受体阻滞剂。
- GC13085 Terazosin A potent and selective α1-AR antagonist
- GC61320 Terazosin dimer impurity dihydrochloride Terazosindimerimpuritydihydrochloride是Terazosin的二聚体,也是Terazosin的杂质。Terazosin是喹唑啉衍生物,是竞争性的,具有口服活性的α1-肾上腺素(α1-adrenoceptor)受体拮抗剂。
- GC13993 Terazosin HCl A potent and selective α1-AR antagonist
- GC50017 Terazosin hydrochloride A potent and selective α1-AR antagonist
- GC11211 Terbutaline Sulfate An Analytical Reference Standard
- GC32637 Tertatolol ((±)-Tertatolol) Tertatolol ((±)-Tertatolol) 是一种有效的 β-肾上腺素受体和 5-HT 受体拮抗剂,具有独特的肾血管扩张作用。
- GC39016 Tetrahydroalstonine Tetrahydroalstonine 是从 Rhazya stricta 的果实中分离出来的吲哚生物碱,是选择性的 α2-肾上腺素受体拮抗剂。
- GC14962 Tetrahydrozoline HCl An α1-adrenergic receptor agonist
- GC12468 Timolol Maleate A non-selective β-adrenergic receptor antagonist
- GC31150 Tiodazosin (BL-5111) Tiodazosin (BL-5111) 是一种有效的竞争性突触后 α 肾上腺素受体拮抗剂。
- GC15629 Tizanidine An α2-adrenergic receptor agonist
- GC17891 Tizanidine HCl An α2-adrenergic receptor agonist
- GC63310 Tizanidine-d4 An internal standard for the quantification of tizanidine
- GC32574 Todralazine (Ecarazine) Todralazine (Ecarazine) (Ecarazine) 是一种抗高血压剂,作为 β2AR 阻滞剂,具有抗氧化和自由基清除活性。
- GC18327 Todralazine (hydrochloride) A β2-adrenergic receptor antagonist
- GC30405 Tolazoline (Imidaline) Tolazoline (Imidaline)(Imidaline) 是一种非选择性竞争性 α-adrenergic receptor 拮抗剂。
- GC18092 Tolazoline HCl An α1- and α2-adrenergic receptor antagonist
- GC13031 Trifluoperazine 2HCl An anti-adrenergic and anti-dopaminergic agent
- GC63241 Trifluoperazine D8 Trifluoperazine D8 是 Trifluoperazine 的氘代物。Trifluoperazine 是一种抗精神病药物吩噻嗪类药物,是一种选择性的 α1-肾上腺素能受体拮抗剂。Trifluoperazine 也是一种有效的多巴胺 D2 受体抑制剂。