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Home >> Signaling Pathways >> Endocrinology and Hormones >> Androgen Receptor

Androgen Receptor(雄激素受体)

AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.

Products for  Androgen Receptor

  1. Cat.No. 产品名称 Information
  2. GC32402 ORM-15341 ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 value of 38 nM and the inhibition constant (Ki) value of 8?nM.
  3. GC31742 Ailanthone (δ13-Dehydrochaparrinone)

    臭椿酮,Δ13-Dehydrochaparrinone

     A quassinoid with diverse biological activities
  4. GC31738 ACP-105 ACP-105 is an orally available and potent selective androgen receptor modulator (SARM) with pEC50 of 9.0 and 9.4 for AR wild type and AR mutation T877A, respectively.
  5. GC31577 Bifluranol (BX341)

    BX341

    Bifluranol (BX341) (BX341) 是一种抗雄激素。
  6. GC31442 YK11 A partial agonist of the androgen receptor
  7. GC31441 DJ-V-159 DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A).
  8. GC31380 LY2452473 LY2452473是一种口服生物可利用的选择性雄激素受体(androgenreceptor)调节剂(SARM)。
  9. GC31254 Androst-4-ene-3,17-diol, dipropanoate, (3β,17β)- (Androst-4-ene-3β,17β-diol, dipropionate)

    Androst-4-ene-3,17-diol,dipropanoate,(3β,17β)-是睾酮代谢物4-雄烯二醇的二丙酸酯。
  10. GC30710 (R)-UT-155 (R)-UT-155(compound11)是一种选择性的、雄激素受体降解物(SARD)配体。活性低于S型异构体。
  11. GC30101 GLPG0492 R enantiomer GLPG0492Renantiomer是GLPG0492的R型对映体，GLPG0492是新型选择性SARM
  12. GC30086 GLPG0492 A selective androgen receptor modulator
  13. GC19458 6β-hydroxy Testosterone

    6-B-羟基-17Β-羟基-4-烯-3-酮丙酸酯,4-Androsten-6β,17β-diol-3-one, 6β, 17β,-Dihydroxyandrost-4-en-3-one

    CYP3A metabolite of testosterone
  14. GC19305 RAD140

    RAD140

     An androgen receptor modulator
  15. GC18496 Leelamine (hydrochloride)

    脱氢松香胺盐酸盐

     An inhibitor of pyruvate dehydrogenase kinase
  16. GC17679 GSK2881078 A selective androgen receptor modulator
  17. GC17160 2-hydroxy Flutamide

    羟基氟他胺,Hydroxyniphtholide,SCH 16423

     An active metabolite of the antiandrogen flutamide
  18. GC15774 5α-dihydro-11-keto Testosterone

    17BETA-羟基-5ALPHA-雄甾烷-3,11-二酮,5α-Androstane-3,11-dione-17β-ol,11-keto Dihydrotestosterone,17β-hydroxy-5α-Androstane-3,11-dione

     An Analytical Reference Standard
  19. GC10785 Danazol

    达那唑

     An androgen receptor agonist
  20. GC14221 HE-3235

    Apoptone,17α-Ethynyl-5α-androstane-3α,17ß-diol

     Androgen receptor antagonist
  21. GC11957 RD162

    N-甲基-4-[7-(4-氰基-3-三氟甲基苯基)-8-氧代-6-硫酮-5,7-二氮杂螺[3.4]辛烷-5-基]-2-氟苯甲酰胺

     A second-generation androgen receptor antagonist
  22. GC11837 MI-136 A menin-MLL inhibitor
  23. GC10618 Fluoxymesterone

    氟甲睾酮

     An Analytical Reference Standard
  24. GC16631 EPI-001

    双酚A

     An androgen receptor antagonist
  25. GC11386 ODM-201

    达洛鲁胺,ODM-201; BAY-1841788

     An androgen receptor antagonist
  26. GC12445 TFM-4AS-1 androgen receptor modulator
  27. GC14560 Cl-4AS-1 Cl-4AS-1 是一种有效的甾体雄激素受体 (AR) 激动剂 (IC50 = 12 nM)，也是 5α-还原酶 I 型和 II 型的抑制剂（IC50 分别为 6 和 10 nM）。
  28. GC17491 CITCO An agonist of human CAR
  29. GC10567 TCPOBOP An agonist for mouse CAR
  30. GC12938 PF 998425 A non-steroidal androgen receptor antagonist
  31. GC12974 Medroxyprogesterone acetate

    醋酸甲羟孕酮; Medroxyprogesterone 17-acetate; Farlutin

     Medroxyprogesterone acetate（MPA）是一种人工合成的孕激素。
  32. GC12516 Spironolactone

    螺内酯; SC9420

     An Analytical Reference Standard
  33. GC12126 Flutamide

    氟他胺; SCH 13521

     An androgen receptor antagonist and a prodrug form of 2-hydroxy flutamide
  34. GC11796 Estradiol valerate

    戊酸雌二醇,β-Estradiol 17-valerate

     A synthetic estrogen
  35. GC13072 Epiandrosterone

    表雄酮; 3β-Androsterone; trans-Androsterone; iso-Androsterone

     An Analytical Reference Standard
  36. GC11070 Dehydroepiandrosterone (DHEA)

    脱氢表雄酮; Prasterone; Dehydroisoandrosterone; Dehydroepiandrosterone

     脱氢表雄酮 (DHEA) 及其硫酸酯 DHEAS 共同代表了人体内最丰富的类固醇激素。
  37. GC13362 TOK-001

    TOK-001; VN-124-1

     A CYP17 inhibitor
  38. GC13971 Cyproterone Acetate

    醋酸环丙孕酮

     An androgen receptor antagonist
  39. GC16840 ARN-509

    阿帕鲁胺,ARN 509; ARN509, Apalutamide

     ARN-509是一种合成的双芳基硫代乙内酰脲化合物，抑制雄激素受体（AR），IC50值为16nM。
  40. GC10372 AZD3514 A SARD
  41. GC13685 Andarine

    S-4

     A selective androgen receptor modulator
  42. GC12271 Bicalutamide

    比卡鲁胺

     A non-steroidal antiandrogen
  43. GC12933 RU 58841

    RU58841; RU-58841

     A non-steroidal antiandrogen
  44. GC10547 ASC-J9

    二甲基姜黄素,GO-Y025; Dimethylcurcumin; ASC J9; GO Y025

     A selective enhancer of AR degradation
  45. GC12791 3,3'-Diindolylmethane

    3,3'-二吲哚甲烷,diindolylmethane, 3,3'-Methylenediindole,DIM,Arundine,HB236

     A phytochemical with antiradiation and chemopreventative effects
  46. GC17557 17 alpha-propionate

    克拉司酮,17α-propionate; CB-03-01

     A peripherally selective androgen receptor antagonist
  47. GC16649 TAK-700 (Orteronel) A non-steroidal inhibitor of the 17,20-lyase activity of CYP17A1
  48. GC12385 MDV3100 (Enzalutamide)

    恩杂鲁胺; MDV3100

     MDV3100(enzalutamide) 是第二代 AR 拮抗剂，在 LNCaP 前列腺细胞中的 IC50 为 36nM。
  49. GN10268 Triptophenolide

    雷酚内酯; Hypolide; (+)-Triptophenolide

     A diterpenoid with antiandrogenic activity
  50. GN10142 Lupeol

    羽扇豆醇; Clerodol; Monogynol B; Fagarasterol

     A dietary triterpene with anti-inflammatory and anticancer activity

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