Rho
Rho GTPases act as molecular switches that convert and amplify external signals into cellular effects upon activation of cell surface receptor in various signaling transduction pathway. It functions in cell proliferation, motility, survival cytoskeletal remodeling and membrane trafficking etc.
- Cat.No. 产品名称 Information
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GC14497
(S)-CCG-1423
A stereoisomer of CCG-1423, a Rho inhibitor
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GC10419
(R)-CCG-1423
A stereoisomer of CCG-1423, a Rho inhibitor
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GC14986
CCG-100602
A Rho/MKL1 transcriptional pathway inhibitor
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GC12795
CCG-1423
An inhibitor of Rho-mediated cell signalling
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GC12817
K–115 hydrochloride dihydrate
K-115 hydrochloride dihydrate (K-115) 是 ROCK 的特异性抑制剂,对 ROCK2 和 ROCK1 的 IC50 分别为 19 和 51 nM。
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GC15478
6H05
An allosteric inhibitor of oncogenic K-Ras(G12C)
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GC11754
AS 1892802
A ROCK1 and ROCK2 inhibitor
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GC15170
SB 772077B dihydrochloride
A ROCK1 and ROCK2 inhibitor
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GC17388
K-Ras(G12C) inhibitor 6
K-Ras(G12C) inhibitor 6 是一种不可逆的 K-Ras(G12C) 变构抑制剂。
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GC10030
EHop-016
A Rac1 and Rac3 inhibitor
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GC12470
ZCL278
A selective Cdc42 inhibitor
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GC10069
NSC 23766 trihydrochloride
Inhibitor of Rac1
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GC14701
Zoledronic Acid
A bisphosphonate that inhibits bone resorption