Trk(酪氨酸激酶)
Trk is a family of tyrosine kinases that regulates synaptic strength and plasticity in the mammalian nervous system.
- Cat.No. 产品名称 Information
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GC65009
PF-6683324
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GC62597
DS-1205b free base
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GC50660
HIOC
HIOC 是 TrkB(原肌球蛋白相关激酶 B)受体的有效和选择性激活剂。
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GC60372
TrkA-IN-1
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GC50346
PF 06273340
PF 06273340 是一种有效的、选择性的、口服生物可利用的和外周受限的 pan Trk 抑制剂。
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GC36425
LOXO-101 (Larotrectinib)
A pan-Trk inhibitor
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GC33112
CH7057288
CH7057288 is a potent and selective TRK inhibitor with IC50 values of 1.1 nM, 7.8 nM and 5.1 nM for TRKA, TRKB, and TRKC respectively.
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GC33090
AZ-23 (AZ23)
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GC32808
Selitrectinib (LOXO-195)
A Trk kinase inhibitor
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GC32623
CE-245677
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GC31676
Tavilermide (MIM-D3)
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GC30770
LM22B-10
An activator of TrkB and TrkC
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GC19362
Repotrectinib
A multi-kinase inhibitor
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GC19332
Sitravatinib
A multi-kinase inhibitor
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GC19063
Belizatinib
An ALK inhibitor
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GC19012
(R)-GNE-140
(R)-GNE-140 是一种有效的乳酸脱氢酶 A (LDHA) 抑制剂,对 LDHA 和 LDHB 的 IC50 分别为 3 nM 和 5 nM; (R)-GNE-140 的效力是 S 对映体的 18 倍。
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GC15365
N-Acetylserotonin
The immediate precursor of melatonin
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GC15282
LOXO-101 (Larotrectinib) sulfate
A pan-Trk inhibitor
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GC14476
Entrectinib
A pan-Trk, ROS1, and ALK inhibitor
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GC16604
Altiratinib
A multiple kinase inhibitor
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GC17622
Ro 08-2750
A p75NTR ligand
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GC11486
ANA 12
A TrkB receptor antagonist
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GC17835
LM 22A4
An agonist of TrkB
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GC16853
7,8-Dihydroxyflavone
A TrkB kinase inhibitor
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GC13780
Cyclotraxin B
Cyclotraxin B 是一种环状肽,是一种高效的选择性 TrkB 抑制剂,不会改变 BDNF 的结合。
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GC12186
BDNF (human)
activator of TrkB and p75 neurotrophin receptors
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GC10720
NTR 368
NTR 368 是衍生自 p75 神经营养因子受体 (p75NTR) 的肽,对应于人类受体的 368-381 位残基。
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GC11362
K 252a
A non-selective PKC inhibitor
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GC15271
Tyrphostin AG 879
A non-specific tyrphostin ErbB2 inhibitor
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GC14123
GW441756
A potent inhibitor of TrkA
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GC16343
GNF-5837
A pan-Trk inhibitor
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GC17033
Lestaurtinib
A potent JAK2 and PRK1 kinase inhibitor
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GC11496
TLQP 21
TLQP 21 是一种 VGF 衍生肽,具有内分泌和内分泌特性,是一种有效的 G 蛋白偶联受体补体 3a 受体 1 (C3aR1) 激动剂(EC50:小鼠 TLQP 21\u003d10.3 μM;人 TLQP 21\u003d68.8 μM) .