Drug Metabolite(药物代谢物)
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
Products for Drug Metabolite
- Cat.No. 产品名称 Information
- GC49421 Atorvastatin lactone-d5 An internal standard for the quantification of atorvastatin lactone
- GC49410 CVT-2738 An active metabolite of ranolazine
- GC49409 Desmethyl Ranolazine A metabolite of ranolazine
- GC49406 ACT-373898 A metabolite of macitentan
- GC49403 Benzarone An active metabolite of benzbromarone
- GC49399 N-Desbutyl Dronedarone (hydrochloride) An active metabolite of dronedarone
- GC49391 7α-Thiospironolactone An active metabolite of spironolactone
- GC49367 4’-hydroxy Atomoxetine Glucuronide (hydrate) A metabolite of atomoxetine
- GC49366 1-Salicylate Glucuronide A metabolite of salicylic acid and aspirin
- GC49365 25-Desacetyl Rifampicin A major active metabolite of rifampicin
- GC49363 Salicyluric Acid A major metabolite of aspirin and salicylic acid
- GC49355 Norfluoxetine-d5 (hydrochloride) An internal standard for the quantification of norfluoxetine
- GC49349 O-Desethyl Sildenafil A metabolite of sildenafil
- GC49340 Pitavastatin lactone-d4 An internal standard for the quantification of pitavastatin lactone
- GC49337 4-Acetamidobenzenesulfonamide A metabolite of asulam and sulfanilamide
- GC49330 2-(2-Aminoethyl)-3-(4-chlorophenyl)-3-hydroxyisoindol-1-one (hydrochloride) A metabolite of mazindol
- GC49316 O-Desmethyl-N-deschlorobenzoyl Indomethacin A metabolite of indomethacin
- GC49315 5-hydroxy Indomethacin A metabolite of indomethacin
- GC49298 7α-Thiomethylspironolactone A major metabolite of spironolactone
- GC49294 1-(4-Chlorobenzhydryl)piperazine An inactive metabolite of meclizine and chlorcyclizine
- GC49291 rac-N-desmethyl Ivabradine-d6 (hydrochloride) An internal standard for the quantification of N-desmethyl ivabradine
- GC49289 Dolutegravir O-β-D-Glucuronide A metabolite of dolutegravir
- GC49288 Dolutegravir M1 A metabolite of dolutegravir
- GC49282 Hydroxy Lenalidomide A metabolite of lenalidomide
- GC49256 N-acetyl Lenalidomide A metabolite of lenalidomide
- GC49252 4’-hydroxy Trazodone A metabolite of trazodone
- GC49250 Hydroxydehydro Nifedipine Carboxylate A metabolite of nifedipine
- GC49241 Methyl Diethyldithiocarbamate An active metabolite of disulfiram
- GC49235 6-Methylmercaptopurine A metabolite of 6-mercaptopurine
- GC49219 N-desmethyl Eletriptan A metabolite of eletriptan
- GC49218 Imidafenacin Metabolite M4 A metabolite of imidafenacin
- GC49217 Trifluoperazine N-Glucuronide A metabolite of trifluoperazine
- GC49216 ADL 08-0011 (hydrochloride) An active metabolite of alvimopan
- GC49213 trans-hydroxy Glimepiride An active metabolite of glimepiride
- GC49212 trans-carboxy Glimepiride A metabolite of glimepiride
- GC49211 O-desmethyl Brinzolamide (hydrochloride) An active metabolite of brinzolamide
- GC49210 N-desethyl Brinzolamide (oxalate) An active metabolite of brinzolamide
- GC49203 rac-Desethyl Oxybutynin (hydrochloride) An active metabolite of oxybutynin
- GC49202 Desmethyl Mirtazapine (hydrochloride) A metabolite of mirtazapine
- GC49189 (E/Z)-4-hydroxy Tamoxifen-d5 An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen
- GC49186 O-Demethyl Apremilast An active metabolite of apremilast
- GC49185 Mirtazapine N-oxide A metabolite of mirtazapine
- GC49184 Palonosetron N-oxide A metabolite of palonosetron
- GC49179 (S)-O-Desmethyl Naproxen A metabolite of (S)-naproxen
- GC49174 Desmethyl Bosentan An active metabolite of bosentan
- GC49173 N-Despropyl Ropinirole An active metabolite of ropinirole
- GC49159 2-(1-Piperazinyl)pyrimidine An α2-AR antagonist and active metabolite of azapirones
- GC49157 rac-5-carboxy Tolterodine An inactive metabolite of tolterodine
- GC49156 Etodolac Acyl Glucuronide A phase II metabolite of etodolac
- GC49152 Celecoxib Carboxylic Acid An inactive metabolite of celecoxib