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Drug Metabolite(药物代谢物)

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Products for  Drug Metabolite

  1. Cat.No. 产品名称 Information
  2. GC49421 Atorvastatin lactone-d5 An internal standard for the quantification of atorvastatin lactone
  3. GC49410 CVT-2738 An active metabolite of ranolazine
  4. GC49409 Desmethyl Ranolazine A metabolite of ranolazine
  5. GC49406 ACT-373898 A metabolite of macitentan
  6. GC49403 Benzarone An active metabolite of benzbromarone
  7. GC49399 N-Desbutyl Dronedarone (hydrochloride) An active metabolite of dronedarone
  8. GC49391 7α-Thiospironolactone An active metabolite of spironolactone
  9. GC49367 4’-hydroxy Atomoxetine Glucuronide (hydrate) A metabolite of atomoxetine
  10. GC49366 1-Salicylate Glucuronide A metabolite of salicylic acid and aspirin
  11. GC49365 25-Desacetyl Rifampicin A major active metabolite of rifampicin
  12. GC49363 Salicyluric Acid A major metabolite of aspirin and salicylic acid
  13. GC49355 Norfluoxetine-d5 (hydrochloride) An internal standard for the quantification of norfluoxetine
  14. GC49349 O-Desethyl Sildenafil A metabolite of sildenafil
  15. GC49340 Pitavastatin lactone-d4 An internal standard for the quantification of pitavastatin lactone
  16. GC49337 4-Acetamidobenzenesulfonamide A metabolite of asulam and sulfanilamide
  17. GC49330 2-(2-Aminoethyl)-3-(4-chlorophenyl)-3-hydroxyisoindol-1-one (hydrochloride) A metabolite of mazindol
  18. GC49316 O-Desmethyl-N-deschlorobenzoyl Indomethacin A metabolite of indomethacin
  19. GC49315 5-hydroxy Indomethacin A metabolite of indomethacin
  20. GC49298 7α-Thiomethylspironolactone A major metabolite of spironolactone
  21. GC49294 1-(4-Chlorobenzhydryl)piperazine An inactive metabolite of meclizine and chlorcyclizine
  22. GC49291 rac-N-desmethyl Ivabradine-d6 (hydrochloride) An internal standard for the quantification of N-desmethyl ivabradine
  23. GC49289 Dolutegravir O-β-D-Glucuronide A metabolite of dolutegravir
  24. GC49288 Dolutegravir M1 A metabolite of dolutegravir
  25. GC49282 Hydroxy Lenalidomide A metabolite of lenalidomide
  26. GC49256 N-acetyl Lenalidomide A metabolite of lenalidomide
  27. GC49252 4’-hydroxy Trazodone A metabolite of trazodone
  28. GC49250 Hydroxydehydro Nifedipine Carboxylate A metabolite of nifedipine
  29. GC49241 Methyl Diethyldithiocarbamate An active metabolite of disulfiram
  30. GC49235 6-Methylmercaptopurine A metabolite of 6-mercaptopurine
  31. GC49219 N-desmethyl Eletriptan A metabolite of eletriptan
  32. GC49218 Imidafenacin Metabolite M4 A metabolite of imidafenacin
  33. GC49217 Trifluoperazine N-Glucuronide A metabolite of trifluoperazine
  34. GC49216 ADL 08-0011 (hydrochloride) An active metabolite of alvimopan
  35. GC49213 trans-hydroxy Glimepiride An active metabolite of glimepiride
  36. GC49212 trans-carboxy Glimepiride A metabolite of glimepiride
  37. GC49211 O-desmethyl Brinzolamide (hydrochloride) An active metabolite of brinzolamide
  38. GC49210 N-desethyl Brinzolamide (oxalate) An active metabolite of brinzolamide
  39. GC49203 rac-Desethyl Oxybutynin (hydrochloride) An active metabolite of oxybutynin
  40. GC49202 Desmethyl Mirtazapine (hydrochloride) A metabolite of mirtazapine
  41. GC49189 (E/Z)-4-hydroxy Tamoxifen-d5 An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen
  42. GC49186 O-Demethyl Apremilast An active metabolite of apremilast
  43. GC49185 Mirtazapine N-oxide A metabolite of mirtazapine
  44. GC49184 Palonosetron N-oxide A metabolite of palonosetron
  45. GC49179 (S)-O-Desmethyl Naproxen A metabolite of (S)-naproxen
  46. GC49174 Desmethyl Bosentan An active metabolite of bosentan
  47. GC49173 N-Despropyl Ropinirole An active metabolite of ropinirole
  48. GC49159 2-(1-Piperazinyl)pyrimidine An α2-AR antagonist and active metabolite of azapirones
  49. GC49157 rac-5-carboxy Tolterodine An inactive metabolite of tolterodine
  50. GC49156 Etodolac Acyl Glucuronide A phase II metabolite of etodolac
  51. GC49152 Celecoxib Carboxylic Acid An inactive metabolite of celecoxib

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