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Home >> Signaling Pathways >> MAPK Signaling >> MEK1/2

MEK1/2

MEK1/2, also known as MAPKK (mitogen-activated protein kinase kinase), is a kinase enzyme which phosphorylates MAPK (mitogen-activated protein kinase).

  1. Cat.No. 产品名称 Information
  2. GC64904 MAP855
  3. GC64292 MS432
  4. GC63554 PD0325901-O-C2-dioxolane
  5. GC63264 Zapnometinib Zapnometinib (PD0184264, ATR-002), an major active metabolite of CI-1040, is a novel MEK inhibitor with an IC50 of 5.7 nM.
  6. GC38653 Selumetinib sulfate
  7. GC37523 RGB-286638 free base A multi-kinase inhibitor
  8. GC37522 RGB-286638 A multi-kinase inhibitor
  9. GC37516 Refametinib R enantiomer
  10. GC36199 GW284543 GW284543 (UNC10225170), a MEK5-selective inhibitor, inhibits MEK5 in a dose-dependently way as determined by reductions in pERK5, and decreases endogenous MYC protein.
  11. GC35719 Cobimetinib hemifumarate A potent, orally available MEK1 inhibitor
  12. GC35684 CHMFL-EGFR-202
  13. GC45099 U-0126

    A MEK inhibitor and AMPK activator
  14. GC43885 Hypothemycin A resorcylic acid lactone polyketide with diverse biological activities
  15. GC41573 Theaflavin 3,3'-digallate A polyphenol with diverse biological activities
  16. GC33831 Lidocaine hydrochloride (Lignocaine hydrochloride) An Analytical Reference Standard
  17. GC33388 MEK-IN-1
  18. GC33305 Balamapimod (MKI 833)
  19. GC30162 trans-Zeatin

    A cytokinin plant growth regulator
  20. GC15646 PD 184161 A potent MEK1/2 inhibitor
  21. GC15240 APS-2-79 An inhibitor of KSR-dependent MAPK signaling
  22. GC17828 BI-847325 A selective dual MEK/Aurora kinase inhibitor
  23. GC14647 SCH772984 HCl

    A selective inhibitor of ERK1/2
  24. GC15044 SCH772984 TFA

    A selective inhibitor of ERK1/2
  25. GC12406 RO5126766(CH5126766) A dual inhibitor of MEK1 and Raf kinases
  26. GC12006 GDC-0994 A selective ERK1/2 inhibitor
  27. GC17485 PD 334581 A MEK inhibitor
  28. GC12851 10Z-Hymenialdisine A natural alkaloid that inhibits MEK-1 and other kinases
  29. GC17964 PD 198306 A potent inhibitor of MEK1/2
  30. GC15061 U0124 An inactive analog of U-0126
  31. GC14247 GDC-0623 A potent, ATP-uncompetitive inhibitor of MEK1
  32. GC16872 Refametinib An allosteric inhibitor of MEK1/2
  33. GC10209 TAK-733 A MEK1 inhibitor
  34. GC12141 RO4987655 A MEK inhibitor
  35. GC14643 AZD8330 A MEK1/2 inhibitor
  36. GC12843 MEK162 (ARRY-162, ARRY-438162) A MEK1/2 inhibitor
  37. GC15693 BIX 02188 A potent MEK5 inhibitor
  38. GC12220 BIX 02189 An inhibitor of MEK5 and ERK5
  39. GC10110 PD318088 An allosteric inhibitor of MEK1
  40. GC18050 Pimasertib (AS-703026) A MEK1/2 inhibitor
  41. GC12989 PD184352 (CI-1040) A potent MEK inhibitor
  42. GC15359 SL-327 A selective MEK1/2 inhibitor
  43. GC12819 PD98059

    A MAPK pathway inhibitor and AMPK activator
  44. GC17608 Lidocaine An Analytical Reference Standard
  45. GC17030 AZD6244(Selumetinib) A highly selective inhibitor of MEK1/2
  46. GC15260 Trametinib DMSO solvate Trametinib DMSO solvate (GSK-1120212 (DMSO solvate);JTP-74057 (DMSO solvate)) 是一种具有口服活性的 MEK 抑制剂，抑制 MEK1 和 MEK2，IC50 约为 2 nM。 Trametinib DMSO solvate 激活自噬并诱导细胞凋亡。
  47. GC16001 SCH772984

    A selective inhibitor of ERK1/2
  48. GC11277 MEK inhibitor MEK 抑制剂是一种有效的 MEK 抑制剂，具有抗肿瘤效力。
  49. GC14337 Cobimetinib (R-enantiomer) Cobimetinib R-对映异构体是 Cobimetinib 活性较低的 R-对映异构体。 Cobimetinib 是一种有效的选择性 MEK 抑制剂。
  50. GC17426 Cobimetinib (racemate) Cobimetinib（消旋体）（GDC-0973 消旋体；XL518 消旋体）是 Cobimetinib 的消旋体。 Cobimetinib 是一种有效的选择性 MEK 抑制剂。
  51. GC10033 Cobimetinib A potent, orally available MEK1 inhibitor

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