NMDA Receptor(NMDA受体)

NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.

Products for NMDA Receptor

Cat.No. 产品名称 Information
GC11335 DL-AP7 DL-AP7 是一种竞争性 NMDA 拮抗剂和抗惊厥药。
GC13714 Conantokin G Conantokin G 是一种 17 个氨基酸的肽，是一种有效的、选择性的和竞争性的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂。
GC11585 TCN 237 dihydrochloride TCN 237 dihydrochloride 是一种有效的 NR2B 选择性 NMDA 拮抗剂，Ki 为 0.85 nM； NR2B Ca2+ 内流 IC50 为 9.7 nM；对 NR2A、NR2C、NR2D、hERG 通道和 α1-肾上腺素能受体无活性。
GC14121 GLYX 13 A partial agonist of the NMDA receptor
GC12785 ZD 9379 ZD 9379 是一种有效的、具有口服活性的脑渗透性完全拮抗剂，作用于 NMDA 受体的甘氨酸位点。
GC12944 Conantokin-R non-competitive NMDA receptor antagonist
GC15156 Conantokin-T Non-competitive NMDA receptor antagonist
GC16240 MNI-caged-NMDA
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group
GC10043 D-CPP-ene NMDA antagonist
GC10866 Spermidine trihydrochloride An endogenous polyamine
GC11064 Spermine tetrahydrochloride A natural polyamine
GC16915 (2R,3S)-Chlorpheg NMDA receptor antagonist
GC14470 Arcaine sulfate An NMDA receptor antagonist
GC17652 N-(4-Hydroxyphenylacetyl)spermine NMDA receptor antagonist
GC11715 Ibotenic acid An excitotoxic NMDA and metabotropic glutamate receptor agonist
GC11286 ACBC ACBC 是一种 NMDA 受体部分激动剂，作用于甘氨酸位点 NR1。
GC14547 Quinolinic acid An excitotoxic agonist at NMDA receptors
GC17823 L-Cysteinesulfinic acid L-半胱氨酸亚磺酸是几种大鼠代谢型谷氨酸受体 (mGluR) 的有效激动剂，对 mGluR1、mGluR5、mGluR2、mGluR4、mGluR6 和 mGluR8 的 pEC50 分别为 3.92、4.6、3.9、2.7、4.0 和 3.94 .
GC15363 Felbamate hydrate An inhibitor of NMDA receptors and a modulator of GABA_A receptors
GC10522 Felbamate An inhibitor of NMDA receptors and a modulator of GABA_A receptors
GC11470 Flupirtine maleate An activator of Kv7 channels
GC14039 MDL-29951 An NMDA receptor antagonist and GPR17 agonist
GC15270 (-)-MK 801 An NMDA receptor antagonist
GC16986 SDZ 220-581 hydrochloride SDZ 220-581 hydrochloride 是一种口服有效的竞争性 NMDA 受体拮抗剂，pKi 值为 7.7。
GC18118 SDZ 220-581 SDZ 220-581 是一种具有口服活性、强效、竞争性 NMDA 受体拮抗剂，pKi 值为 7.7。
GC16616 (+)-MK 801 强效 NMDA 拮抗剂