GABA Receptor(γ-氨基丁酸受体)
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
Products for GABA Receptor
- Cat.No. 产品名称 Information
- GC15226 SKF 89976A hydrochloride SKF 87699A hydrochloride 是一种选择性 GABA 转运蛋白 (GAT-1) 抑制剂,对 CHO 细胞中的 GAT-1、GAT-2 和 GAT-3 的 IC50 分别为 0.28 μM、137.34 μM 和 202.8 μM。
- GC10183 TPMPA A selective GABAA-ρ1 (ρ1 GABAC) receptor antagonist
- GC16311 Chlormethiazole hydrochloride A potentiator of GABAA receptors
- GC12169 NCS-382 A GHB receptor antagonist
- GC16495 GBLD 345 GABAA receptor agonist
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GC16569
PK 11195
A high affinity ligand for peripheral benzodiazepine receptor, TSPO
- GC16238 FGIN-1-43 ligand as probe for the mitochondial DBI receptor (peripheral benzodiazepine receptor)
- GC14017 FGIN-1-27 A TSPO agonist
- GC17381 trans-4-Hydroxycrotonic acid ligand of γ-hydroxybutyric acid (GHB) receptor
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GC11449
β-CCB
benzodiazepine receptor ligand
- GC12506 3-Methyl-GABA 3-Methyl-GABA 是一种有效的 GABA 氨基转移酶激活剂。
- GC14942 SKF 97541 GABAB激动剂
- GC17257 Saclofen A GABAB receptor antagonist
- GC11267 2-Hydroxysaclofen 2-Hydroxysaclofen 是一种有效的 γ-amino-butyric-acid-B (GABAB) 受体拮抗剂。
- GC10967 TACA An agonist of homomeric GABAA receptors
- GC10313 ZAPA sulfate GABAA receptors agonist
- GC17691 Phaclofen Phaclofen 是一种选择性 GABAB 受体拮抗剂。
- GC15636 (-)-Bicuculline methochloride An enantiomer of (+)-bicuculline methochloride
- GC16857 (-)-Bicuculline methobromide (-)-Bicuculline methobromide (l-Bicuculline methobromide) 是一种有效的 GABAA 受体拮抗剂。
- GC11612 RuBi GABA trimethylphosphine GABAB receptor agonist
- GC17321 RuBi-GABA RuBi-GABA 是一种新型的钌基笼状 GABA 化合物。
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GC14150
DPNI-caged-GABA
activates GABAA receptor
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GC14192
Allopregnanolone
A positive modulator of GABAA receptors
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GC17399
Pregnanolone
GABAA receptor positive allosteric modulator
- GC11565 Bretazenil A positive allosteric modulator of GABAA receptors
- GC11600 Valerenic acid Valerenic acid ((-)-Valerenic Acid) 是一种倍半萜类化合物,是一种具有口服活性的 GABAA 受体正变构调节剂。
- GC12357 Pentylenetetrazole A seizure-inducing compound
- GC12359 Hispidulin A flavonoid with diverse biological activities
- GC10844 SCS GABAA receptor antagonist
- GC10856 THIP hydrochloride A GABAA receptor agonist and GABAC receptor antagonist
- GC12568 FG 7142 A benzodiazepine receptor ligand
- GC10530 Dihydroergotoxine mesylate A mixture of alkaloids with diverse biological activities
- GC14834 (±)-Nipecotic acid A GAT inhibitor
- GC13567 Isoguvacine hydrochloride A GABAA receptor agonist
- GC14659 Guvacine hydrochloride An inhibitor of GABA uptake
- GC10186 Tiagabine A GAT-1 inhibitor
- GC17402 Tiagabine hydrochloride A GAT-1 inhibitor
- GC13387 Vigabatrin Hydrochloride Inhibitor of GABA transaminase
- GC16564 Niflumic acid A selective COX-2 inhibitor
- GC15960 Primidone An Analytical Reference Material
- GC16691 Chlormezanone A muscle relaxant
- GC11901 Nefiracetam An Analytical Reference Standard
- GC12414 Bemegride Bemegride (3-Ethyl-3-methylglutarimide) 是一种中枢神经系统兴奋剂和巴比妥类中毒的解毒剂。
- GC13792 Rufinamide An anticonvulsant
- GC14111 (R)-baclofen (R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。
- GC10974 AWD 131-138 A partial agonist of the GABAA receptor
- GC13802 Riluzole Riluzole 是一种抗惊厥药,属于使用依赖性 Na+ 通道阻滞剂家族,它也可以抑制 GABA 摄取,IC50 为 43 μM。
- GC12714 Gabapentin An approved antiepileptic drug
- GC10772 Flumazenil A GABAA receptor antagonist and partial agonist
- GC12599 Retigabine dihydrochloride An Analytical Reference Standard