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GPCR/G protein

  1. Cat.No. Product Name Information
  2. GC12823 (R,S)-Atenolol β1-adrenergic receptor antagonist
  3. GC19541 (rac)-Antineoplaston A10

    (rac)-Antineoplaston A10 is the racemate of Antineoplaston A10

  4. GC38721 (Rac)-E1R (Rac)-E1R (Compound 2) 是 E1R 的外消旋体。(Rac)-E1R 是 sigma-1 受体的正变构调节剂 (Sig1R PAM),可用于治疗认知和记忆障碍。
  5. GC34367 (RS)-Butyryltimolol (RS)-Butyryltimolol是Butyryltimolol的外消旋体。Butyryltimolol是Timolol的丁酸酯。Timolol是非选择性β受体阻滞剂。
  6. GC12279 (RS)-MCPG mGluR antagonist
  7. GC15292 (S)-(+)-Niguldipine hydrochloride L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
  8. GC12463 (S)-(-)-Atenolol β-adrenergic blocker
  9. GC15039 (S)-(-)-Pindolol beta-adrenergic antagonist
  10. GC16637 (S)-(-)-Propranolol hydrochloride β-adrenoceptor antagonist
  11. GC60006 (S)-Carvedilol (S)-Carvedilol 是 Carvedilol 的 S 型异构体,是一种非选择性 β/α-1 受体阻断剂。(S)-Carvedilol 可以抵抗 Doxorubicin (DOX) 的血管或心脏毒性。
  12. GC35002 (S)-Mapracorat (S)-Mapracorat 是一种选择性且活性较小的糖皮质激素受体激动剂。
  13. GC16349 (S)-MCPG mGluR antagonist
  14. GC10753 (S)-SLV 319 CB1 receptor antagonist
  15. GC39249 (S)-Terazosin (S)-Terazosin 是 Terazosin 的有活性的 S 型异构体,也是一种有效的,高亲和力的 α-肾上腺素受体拮抗剂,对 α1a,α1b 和 α1d-肾上腺素受体的 Ki 值分别为 3.91 nM,0.79 nM 和 1.16 nM。(S)-Terazosin 对 α2a,α2B 和 α2c-肾上腺素受体也具有高亲和力,Ki 值分别为 729 nM,3.5 nM 和 46.4 nM。
  16. GC60425 (S)-Verapamil D7 hydrochloride (S)-VerapamilD7hydrochloride((S)-(-)-VerapamilD7hydrochloride)是(S)-Verapamilhydrochloride的一种氘代化合物。(S)-Verapamilhydrochloride(S(-)-Verapamilhydrochloride)通过MRP1抑制白三烯C4(LTC4)和钙黄绿素的转运。(S)-Verapamilhydrochloride导致潜在耐药性肿瘤细胞死亡。
  17. GC60008 (S)-Verapamil hydrochloride (S)-Verapamil hydrochloride (S(-)-Verapamil hydrochloride) 通过 MRP1 抑制白三烯 C4 (LTC4) 和钙黄绿素的转运。(S)-Verapamil hydrochloride 导致潜在耐药性肿瘤细胞死亡。
  18. GA20291 (Sar¹)-Angiotensin II The substitution with Sar at position 1 of angiotensin II resulted in a partial agonistic activity.
  19. GC35011 (Z)-Thiothixene (Z)-Thiothixene 是 serotonergic receptor 的拮抗剂,来自专利 US 20150141345 A1。
  20. GC16663 (±)-4-hydroxy Propranolol (hydrochloride) β1- and β2-adrenergic receptors inhibitor
  21. GC15087 (±)-Talinolol β1-selective adrenoceptor antagonist

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