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Home >> Signaling Pathways >> Endocrinology and Hormones >> Estrogen/progestogen Receptor

Estrogen/progestogen Receptor(雌激素/孕激素受体)

The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.

Products for Estrogen/progestogen Receptor

Cat.No. 产品名称 Information
GC16852 Estropipate A piperazine salt form of estrone 3-sulfate
GC17856 RU 58668 Pure antiestrogen that downregulates estrogen receptor expression
GC15975 α-Estradiol A weak estrogen with neuroprotective effects
GC18003 (R,R)-THC (R,R)-THC 是 ERα 激动剂和 ERβ 拮抗剂，对 ERα 和 ERβ 的 Kis 分别为 9.0 nM 和 3.6 nM。
GC11781 Medroxyprogesterone A progesterone receptor agonist
GC13303 Etonogestrel A steroidal progestin
GC15366 Clomiphene citrate A selective estrogen receptor modulator
GC12974 Medroxyprogesterone acetate A synthetic progestogen
GC11436 Ethisterone A synthetic progestin
GC11822 Erteberel (LY500307) A potent and selective agonist of ERβ
GC15324 Hexestrol A synthetic non-steroidal estrogen receptor ligand
GC12000 Ethynodiol diacetate A synthetic progestogen
GC12182 Estriol An estradiol metabolite produced during pregnancy
GC10139 Estradiol Cypionate A synthetic estrogen
GC16292 Equol An estrogen receptor agonist
GC10245 Bazedoxifene HCl Bazedoxifene HCl (TSE-424 hydrochloride) 是一种具有口服活性、可渗透 BBB 的非甾体选择性雌激素受体调节剂 (SERM)，对 ERα 的 IC50 分别为 23 nM 和 99 nM；和ERβ，分别。盐酸巴多昔芬可用于骨质疏松症的研究。 Bazedoxifene HCl 作为 IL-6/GP130 蛋白质-蛋白质相互作用的抑制剂。 Bazedoxifene HCl 可用于胰腺癌的研究。
GC13297 Altrenogest A synthetic progestin
GC14704 Levonorgestrel A synthetic progestin
GC12379 Drospirenone A synthetic progestogen
GC10017 Gestodene A progestin
GC15578 Dienogest A synthetic progestin and PR agonist
GC13835 Toremifene Citrate A selective estrogen receptor modulator
GC11677 Ulipristal acetate A selective progesterone receptor modulator
GC11669 Tamoxifen Citrate A selective estrogen receptor modulator
GC13350 Raloxifene HCl A selective estrogen receptor modulator
GC11688 Megestrol Acetate A synthetic progestogen
GC10789 XCT790 A selective inverse agonist of ERRα
GC11282 β-Estradiol
The major premenopausal estrogen
GC14385 Estrone A primary, naturally-occurring estrogen
GC12408 Progesterone An endogenous hormone and hormone precursor
GC12148 Ethinyl Estradiol A 17β-estradiol analog
GC18000 Fulvestrant (ICI 182,780)
氟维司汀是一种选择性雌激素受体(ER)拮抗剂。它结合、阻断和降解estrogen receptor(ER)，然后抑制ER介导的转录活性，IC₅₀为9.4 nM。
GC11544 Toremifene 托瑞米芬（Z-托瑞米芬）是一种用于预防骨质疏松症的第二代选择性雌激素受体调节剂（SERM）。
GC16847 Tanaproget Tanaproget (NSP-989) 是一种新型非甾体孕酮受体激动剂，与参考甾体孕激素相比，它可以以更高的相对亲和力与来自各种物种的 PR 结合。
GC17200 Nestoron A synthetic progestin
GC10852 Bazedoxifene acetate A selective estrogen receptor modulator
GC14883 Bazedoxifene Bazedoxifene (TSE-424) 是一种口服的、可渗透 BBB 的非甾体选择性雌激素受体调节剂 (SERM)，对 ERα 和 ERβ 的 IC50 分别为 23 nM 和 99 nM。巴多昔芬可用于骨质疏松症的研究。 Bazedoxifene 还作为 IL-6/GP130 蛋白-蛋白相互作用的抑制剂，可用于胰腺癌的研究。
GC15373 (E)-2-Decenoic acid An unsaturated fatty acid found in royal jelly