Cyclin-Dependent Kinases(细胞周期蛋白依赖性激酶)
Cyclin-dependent kinases is a group of serine/threonine kinases. It is activated by binding to cyclin and participates in the regulation of cell cycle.
- Cat.No. 产品名称 Information
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GC50175
CGP 74514 dihydrochloride
Potent cdk1 inhibitor
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GC15841
Alsterpaullone
A dual CDK and GSK3 inhibitor
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GC16520
Olomoucine
An inhibitor of cyclin-dependent kinases
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GC15215
Iso-Olomoucine
An inactive stereoisomer of olomoucine
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GC14294
Cdk1/2 Inhibitor III
A cell-permeable inhibitor of Cdk1 and Cdk2
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GC11564
Cdk4/6 Inhibitor IV
A cell-permeable inhibitor of Cdk4/6
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GC15607
ON123300
A multi-kinase inhibitor
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GC14002
Bohemine
A Cdk inhibitor
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GC15173
PD 0332991 (Palbociclib)
PD 0332991 (Palbociclib) (PD 0332991) 是一种具有口服活性的选择性 CDK4 和 CDK6 抑制剂,IC50 值分别为 11 和 16 nM。 PD 0332991 (Palbociclib) 具有有效的抗增殖活性,可诱导癌细胞的细胞周期停滞,可用于 HR 阳性和 HER2 阴性乳腺癌和肝细胞癌的研究。
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GC18051
CCT251545 analogue, Compound 51
Potent, Selective, orally bioavailable CDK 8/19 Inhibitor
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GC16420
THZ531
An inhibitor of Cdk12 and Cdk13
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GC14230
K03861
K03861 (K03861) 是一种 II 型 CDK2 抑制剂,Kd 为 8.2 nM。 K03861 (K03861) 通过与活化细胞周期蛋白的结合竞争抑制 CDK2 活性。
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GC16545
GX-674
GX-674 是一种有效的、状态依赖性、异构体选择性电压门控钠通道 1.7 (Nav1.7) 拮抗剂,在 -40 mV 时的 IC50 为 0.1 nM。
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GC13511
THZ2
A Cdk7 inhibitor
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GC12826
AZD-5597
Potent CDK inhibitor
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GC14707
Purvalanol A
A selective inhibitor of cyclin-dependent kinases
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GC12348
Ro 3306
An inhibitor of Cdk1
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GC11971
LY2857785
A Cdk9 inhibitor
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GC17067
LDC000067
A Cdk9 inhibitor
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GC11944
PF 4800567 hydrochloride
A selective CK1ε inhibitor
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GC16413
TMCB
A dual inhibitor of CK2 and ERK8
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GC16429
(R)-DRF053 dihydrochloride
cdk/CK1 inhibitor,potent and ATP-competitive
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GC17150
Ryuvidine
An inhibitor of SETD8
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GC12886
NSC 625987
A Cdk4/cyclin D1 complex inhibitor
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GC11410
Aminopurvalanol A
A selective CDK inhibitor
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GC11634
NSC 693868
A selective inhibitor of Cdk1 and Cdk5
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GC13100
[Ala92]-p16 (84-103)
inhibitor of cyclin-dependent kinase-4 (cdk4)/cyclin D1
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GC13649
Arcyriaflavin A
A CDK4 and CAMKII inhibitor
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GC14182
Kenpaullone
A inhibitor of cyclin-dependent kinase and GSK3β
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GC12642
THZ1 Hydrochloride
A covalent Cdk7 inhibitor
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GC14162
ML167
A selective Clk4 inhibitor
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GC10840
THZ1
A covalent Cdk7 inhibitor
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GC15377
LEE011 succinate
A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
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GC15922
LEE011 hydrochloride
A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
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GC11785
CDK4 inhibitor
An antiproliferative cyclin D1/Cdk4 inhibitor
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GC14974
AMG 925
A dual inhibitor of FLT3 and Cdk4
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GC16000
WHI-P180
A multi-kinase inhibitor
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GC17400
R547
A selective Cdk inhibitor
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GC10842
LEE011
A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
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GC16425
Flavopiridol hydrochloride
An inhibitor of cyclin-dependent kinases
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GC11835
Deferasirox
An iron chelator with anticancer activity
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GC16268
Purvalanol B
A CDK inhibitor
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GC17648
Dinaciclib(SCH727965)
A CDK inhibitor
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GC12865
BMS265246
A cell-permeable inhibitor of Cdk1 and Cdk2
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GC15588
PHA-848125
An inhibitor of Cdks
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GC15421
Palbociclib (PD0332991) Isethionate
Palbociclib (PD 0332991) isethionate 是一种具有口服活性的选择性 CDK4 和 CDK6 抑制剂,IC50 值分别为 11 和 16 nM。 Palbociclib (PD0332991) Isethionate 具有有效的抗增殖活性,可诱导癌细胞的细胞周期停滞,可用于 HR 阳性和 HER2 阴性乳腺癌和肝细胞癌的研究。
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GC12438
AZD-5438
A potent inhibitor of CDKs
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GC17935
PD 0332991 (Palbociclib) HCl
A selective cyclin D kinase 4/6 inhibitor
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GC16822
LY2835219
A dual inhibitor of CDK4 and CDK6
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GC15963
Nu 6027
A CDK and ATR inhibitor