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Home >> Signaling Pathways >> Cell Cycle/Checkpoint >> Cyclin-Dependent Kinases

Cyclin-Dependent Kinases(细胞周期蛋白依赖性激酶)

Cyclin-dependent kinases is a group of serine/threonine kinases. It is activated by binding to cyclin and participates in the regulation of cell cycle.

  1. Cat.No. 产品名称 Information
  2. GC50175 CGP 74514 dihydrochloride Potent cdk1 inhibitor
  3. GC15841 Alsterpaullone A dual CDK and GSK3 inhibitor
  4. GC16520 Olomoucine An inhibitor of cyclin-dependent kinases
  5. GC15215 Iso-Olomoucine An inactive stereoisomer of olomoucine
  6. GC14294 Cdk1/2 Inhibitor III A cell-permeable inhibitor of Cdk1 and Cdk2
  7. GC11564 Cdk4/6 Inhibitor IV A cell-permeable inhibitor of Cdk4/6
  8. GC15607 ON123300 A multi-kinase inhibitor
  9. GC14002 Bohemine A Cdk inhibitor
  10. GC15173 PD 0332991 (Palbociclib) PD 0332991 (Palbociclib) (PD 0332991) 是一种具有口服活性的选择性 CDK4 和 CDK6 抑制剂，IC50 值分别为 11 和 16 nM。 PD 0332991 (Palbociclib) 具有有效的抗增殖活性，可诱导癌细胞的细胞周期停滞，可用于 HR 阳性和 HER2 阴性乳腺癌和肝细胞癌的研究。
  11. GC18051 CCT251545 analogue, Compound 51

    Potent, Selective, orally bioavailable CDK 8/19 Inhibitor
  12. GC16420 THZ531 An inhibitor of Cdk12 and Cdk13
  13. GC14230 K03861 K03861 (K03861) 是一种 II 型 CDK2 抑制剂，Kd 为 8.2 nM。 K03861 (K03861) 通过与活化细胞周期蛋白的结合竞争抑制 CDK2 活性。
  14. GC16545 GX-674 GX-674 是一种有效的、状态依赖性、异构体选择性电压门控钠通道 1.7 (Nav1.7) 拮抗剂，在 -40 mV 时的 IC50 为 0.1 nM。
  15. GC13511 THZ2 A Cdk7 inhibitor
  16. GC12826 AZD-5597

    Potent CDK inhibitor
  17. GC14707 Purvalanol A A selective inhibitor of cyclin-dependent kinases
  18. GC12348 Ro 3306 An inhibitor of Cdk1
  19. GC11971 LY2857785 A Cdk9 inhibitor
  20. GC17067 LDC000067 A Cdk9 inhibitor
  21. GC11944 PF 4800567 hydrochloride A selective CK1ε inhibitor
  22. GC16413 TMCB A dual inhibitor of CK2 and ERK8
  23. GC16429 (R)-DRF053 dihydrochloride cdk/CK1 inhibitor,potent and ATP-competitive
  24. GC17150 Ryuvidine An inhibitor of SETD8
  25. GC12886 NSC 625987 A Cdk4/cyclin D1 complex inhibitor
  26. GC11410 Aminopurvalanol A A selective CDK inhibitor
  27. GC11634 NSC 693868 A selective inhibitor of Cdk1 and Cdk5
  28. GC13100 [Ala92]-p16 (84-103) inhibitor of cyclin-dependent kinase-4 (cdk4)/cyclin D1
  29. GC13649 Arcyriaflavin A A CDK4 and CAMKII inhibitor
  30. GC14182 Kenpaullone A inhibitor of cyclin-dependent kinase and GSK3β
  31. GC12642 THZ1 Hydrochloride A covalent Cdk7 inhibitor
  32. GC14162 ML167 A selective Clk4 inhibitor
  33. GC10840 THZ1 A covalent Cdk7 inhibitor
  34. GC15377 LEE011 succinate A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
  35. GC15922 LEE011 hydrochloride A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
  36. GC11785 CDK4 inhibitor An antiproliferative cyclin D1/Cdk4 inhibitor
  37. GC14974 AMG 925 A dual inhibitor of FLT3 and Cdk4
  38. GC16000 WHI-P180 A multi-kinase inhibitor
  39. GC17400 R547 A selective Cdk inhibitor
  40. GC10842 LEE011 A selective cyclin D1/CDK4 and cyclin D3/CDK6 inhibitor
  41. GC16425 Flavopiridol hydrochloride An inhibitor of cyclin-dependent kinases
  42. GC11835 Deferasirox An iron chelator with anticancer activity
  43. GC16268 Purvalanol B A CDK inhibitor
  44. GC17648 Dinaciclib(SCH727965) A CDK inhibitor
  45. GC12865 BMS265246 A cell-permeable inhibitor of Cdk1 and Cdk2
  46. GC15588 PHA-848125 An inhibitor of Cdks
  47. GC15421 Palbociclib (PD0332991) Isethionate Palbociclib (PD 0332991) isethionate 是一种具有口服活性的选择性 CDK4 和 CDK6 抑制剂，IC50 值分别为 11 和 16 nM。 Palbociclib (PD0332991) Isethionate 具有有效的抗增殖活性，可诱导癌细胞的细胞周期停滞，可用于 HR 阳性和 HER2 阴性乳腺癌和肝细胞癌的研究。
  48. GC12438 AZD-5438 A potent inhibitor of CDKs
  49. GC17935 PD 0332991 (Palbociclib) HCl A selective cyclin D kinase 4/6 inhibitor
  50. GC16822 LY2835219 A dual inhibitor of CDK4 and CDK6
  51. GC15963 Nu 6027 A CDK and ATR inhibitor

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