AChE(乙酰胆碱脂酶)
AChE, also know as acetylcholinesterase, is a hydrolase that hydrolyzes the neurotransmitter acetylcholine.
Products for AChE
- Cat.No. 产品名称 Information
- GC43336 Cyanidin 3-O-β-D-Galactopyranoside (chloride) An anthocyanin flavonoid with antioxidant properties
- GC41774 1,2,3-Trimyristoyl-rac-glycerol A triacylglycerol
- GC40847 Neoeriocitrin A flavonoid with antioxidative and osteogenic activities
- GC34288 Pyridostigmine D6 bromide PyridostigmineD6bromide是Pyridostigmine的氘代化合物标准品。
- GC33684 Pralidoxime chloride (2-PAM chloride) An AChE reactivator
- GC33067 Sophoflavescenol Sophoflavescenol是一种异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50值为0.013μM;同时抑制RLAR,HRAR,BACE1,AChE和BChE,IC50值分别为0.30µM,0.17µM,10.98µM,8.37µM和8.21µM。
- GC32194 Metrifonate (Trichlorfon) Metrifonate是一种不可逆的有机磷乙酰胆碱酯酶抑制剂,用作杀虫剂,控制苍蝇和蟑螂。
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GC31699
Scopoletin (Gelseminic acid)
A natural coumarin
- GC31193 Benactyzine hydrochloride Benactyzine hydrochloride is a centrally acting muscarinic antagonist. It is used as an antidepressant in the treatment of depression and associated anxiety.
- GC31190 Demecarium Bromide (BC-48) Demecarium Bromide (BC-48) (BC-48) 是一种有效的胆碱酯酶抑制剂,表观亲和力 (Kiapp) 为 0.15 μM.
- GC31044 T 82 T82是一种有效的5-HT3拮抗剂和乙酰胆碱酯酶(AChE)的抑制剂,用于阿尔茨海默症的研究。
- GC30908 Drofenine hydrochloride (Hexahydroadiphenine hydrochloride) Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
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GC30856
Protriptyline hydrochloride
A tricyclic antidepressant
- GC30810 Donepezil (E2020) An AChE inhibitor
- GC30446 MHP 133 MHP133是一种多靶点抑制剂,可以抑制AChE的活性,KKi值为69μM;同时抑制毒蕈碱M1和M2受体,5HT4受体和咪唑I2受体。
- GC30290 Neostigmine methyl sulfate A reversible acetylcholinesterase inhibitor
- GC18891 Malathion An organophosphate insecticide
- GC18207 Pitofenone (hydrochloride) An antispasmodic agent
- GC15628 bis(7)-Tacrine A potent acetylcholinesterase inhibitor
- GC15438 Asoxime (chloride) An AChE reactivator
- GC17705 Edrophonium (chloride) An AChE inhibitor
- GC11606 4-Methylbenzylidene camphor A UV blocker with estrogenic effects
- GC15604 Hydroxytacrine (maleate) A major active metabolite of tacrine
- GC15895 Itopride hydrochloride An AChE inhibitor and a prokinetic agent
- GC13474 Garcinol A polyisoprenylated benzophenone with diverse biological activities
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GC17385
KML 29
An inhibitor of MAGL
- GC12937 STF 083010 An inhibitor of IRE1 endonuclease activity
- GC15832 GSK 264220A An endothelial lipase inhibitor
- GC14163 PE 154 PE 154 (Compound 13) 是人乙酰胆碱酯酶 (AChE) 和丁酰胆碱酯酶 (BChE) 的有效荧光抑制剂(IC50s 分别为 280 pM 和 16 nM)。
- GC11617 Pristimerin Potent, selective inhibitor of monoacylglycerol lipase
- GC16974 Ambenonium dichloride Ambenonium (WIN 8077) chloride 是一种具有高亲和力的具有口服活性且可逆的乙酰胆碱酯酶 (AChE) 抑制剂。
- GC15203 Acephate An organophosphate insecticide
- GC13783 Phenserine An AChE inhibitor
- GC12813 Tacrine hydrochloride An AChE and butyrylcholinesterase inhibitor
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GC17391
Physostigmine hemisulfate
毒扁豆碱半硫酸盐 (Eserine hemisulfate) 是一种可逆的乙酰胆碱酯酶 (AChE) 抑制剂。
- GC14400 (-)-Huperzine A A neuroprotective AChE inhibitor
- GC15348 Pyridostigmine Bromide An inhibitor of AChE and BChE
- GC14490 Donepezil HCl An AChE inhibitor
- GC12123 sn-Glycero-3-phosphocholine A nootropic phospholipid
- GC12994 Rivastigmine Tartrate A cholinesterase inhibitor
- GC10267 Rivastigmine A cholinesterase inhibitor
- GC16573 Galanthamine An alkaloid with AChE inhibitory and nAChR potentiating activities
- GN10145 Rhodionin Rhodionin 是从 Rhodiola crenulata 的根中分离出来的,是一种特异性的非竞争性细胞色素 P450 2D6 抑制剂,IC50 为 0.761 μM,Ki 为 0.769 μM。
- GN10716 Epiberberine An alkaloid with diverse biological activities
- GN10155 (+)- Corydaline An alkaloid with diverse biological activities
- GN10654 (+)-Corynoline An isoquinoline alkaloid with diverse biological activities
- GN10616 Timosaponin A3 A natural steroid saponin
- GN10437 Imperatorin A furanocoumarin with diverse biological activities
- GN10352 Isoimperatorin A furanocoumarin that inhibits CYP1A
- GN10578 Polygalacic acid A triterpenoid saponin with antioxidant and neuroprotective activities