Tyrosine Kinase
- Bcr-Abl(66)
- Ack1(3)
- Axl(10)
- ALK(50)
- BMX Kinase(3)
- Broad Spectrum Protein Kinase Inhibitor(10)
- c-FMS(29)
- c-Kit(51)
- c-MET(68)
- c-RET(7)
- CSF-1R(3)
- DDR1/DDR2 Receptor(1)
- EGFR(157)
- EphB4(1)
- FAK(28)
- FGFR(70)
- FLT3(70)
- HER2(19)
- IGF1R(25)
- Insulin Receptor(22)
- IRAK(13)
- ITK(8)
- Lck(1)
- LRRK2(18)
- PDGFR(86)
- PTKs/RTKs(4)
- Pyk2(5)
- ROR(25)
- Spleen Tyrosine Kinase (Syk)(25)
- Src(77)
- Tie-2 (2)
- Trk(31)
- VEGFR(142)
- Kinase(0)
- Discoidin Domain Receptor(9)
- DYRK(14)
- Ephrin Receptor(6)
- RET(21)
- ROS(10)
- TAM Receptor(20)
- Cat.No. Product Name Information
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GC38006
β-Hydroxyisovalerylshikonin
Beta-hydroxyisovalerylshikonin 是一种从Lithospermium radix 中分离出的天然产物,是一种有效的 PTK 抑制剂, 对 EGFR 和 v-Src 受体作用的 IC50 分别为 0.7 μM 和 1 μM。Beta-hydroxyisovalerylshikonin 对多种肿瘤细胞系均有抑制作用,能高效诱导 NCI-H522 和 DMS114 细胞的死亡。
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GC13944
(5Z)-7-Oxozeaenol
TAK1 mitogen-activated protein kinase kinase kinase (MAPKKK) inhibitor
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GC17800
(E)-FeCP-oxindole
VEGFR-2 inhibitor
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GC14729
(R)-Crizotinib
C-MET/ALK inhibitor,potent and ATP-competitve
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GC19012
(R)-GNE-140
A TRK kinase (TKI) inhibitor
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GC13136
(S)-Crizotinib
Potent MTH1 inhibitor
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GC13344
(Z)-FeCP-oxindole
VEGFR-2 inhibitor
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GC12172
1-Naphthyl PP1
Src family kinases inhibitor
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GC34119
1-Naphthyl PP1 hydrochloride (1-NA-PP 1 hydrochloride)
1-NaphthylPP1(1-NA-PP1)盐酸盐是src家族抑制剂,对v-Src,c-Fyn,c-Abl,CDK2和CAMKII的IC50分别为1.0,0.6,0.6,18和22μM。
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GC11696
1-NM-PP1
Pp60c-src inhibitor
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GC35053
123C4
123C4 是一种有效、选择性的,竞争性受体酪氨酸激酶 EPHA4 激动剂,Ki 值为 0.65 μM.
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GC33087
2,4-Pyrimidinediamine with linker
2,4-Pyrimidinediaminewithlinker是专利WO2013055780A1(71页,intermediate2),激酶抑制剂,含linker结构。
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GC33519
2,5-Dihydroxybenzoic acid
2,5-Dihydroxybenzoicacid是苯甲酸的代谢物,也是纤维母细胞生长因子(fibroblastgrowthfactor)的强效抑制剂。
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GC10408
2-D08
Sumoylation inhibitor
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GC33319
2-Keto Crizotinib (PF-06260182)
2-KetoCrizotinib(PF-06260182)是有活性的克唑替尼的内酰胺代谢产物。
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GC12818
4-methyl Erlotinib
EGFR inhibitor
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GC11205
5'-Fluoroindirubinoxime
FMS-like receptor tyrosine kinase-3 (FLT3) inhibitor
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GC16853
7,8-Dihydroxyflavone
Tyrosine kinase receptor B (TrkB) agonist
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GC32992
7-Hydroxy-4-chromone (7-Hydroxychromone)
7-Hydroxychromone是一个Src激酶抑制剂,其IC50值小于300μM。
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GC35209
A 419259
A 419259 是一种广谱的吡咯-嘧啶抑制剂,增强对 Src 家族的选择性,作用于 Src,Lck 和 Lyn,IC50 分别为 9 nM,<3 nM 和 <3 nM。