MAPK Signaling

Products for MAPK Signaling
- ERK(59)
- MEK1/2(60)
- NKCC(5)
- MNK(5)
- PKA(33)
- p38(78)
- Rac(2)
- Raf(56)
- RasGAP (Ras- P21)(1)
- JNK(46)
- cAMP(5)
- Protein Kinase G(2)
- RSK(23)
- Other(4)
- MAPKAPK(1)
- MKK(2)
- KLF(2)
- MAP3K(14)
- MAP4K(8)
- MAPKAPK2 (MK2)(5)
- Mixed Lineage Kinase(4)
- Cat.No. Product Name Information
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GC13944
(5Z)-7-Oxozeaenol
TAK1 mitogen-activated protein kinase kinase kinase (MAPKKK) inhibitor
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GC12851
10Z-Hymenialdisine
Pan kinase inhibitor
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GC35132
4-Hydroxylonchocarpin
4-Hydroxylonchocarpin 是一种查尔酮化合物,来自补骨脂 (Psoralea corylifolia) 提取物。4-Hydroxylonchocarpin 增强 p38 MAPK,JNK 和 ERK 的磷酸化。4-Hydroxylonchocarpin 具有多种药理活性,包括抗菌,抗癌,抗逆转录酶,抗结核,抗疟,抗炎和抗氧化活性。
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GC12834
6-Bnz-cAMP sodium salt
cAMP analog,PKA activator
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GC16929
8-Bromo-cAMP, sodium salt
Cell-permeable cAMP analog that activates PKA
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GC15352
8-CPT-Cyclic AMP (sodium salt)
lipophilic activator of the cyclic-AMP- and cyclic-GMP-dependent protein kinases, PKA and PKG
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GC35242
Actein
Actein 是从 Cimicifuga foetida 的根茎中分离的三萜糖苷。Actein 通过促进 ROS/JNK 活化和钝化人膀胱癌中的 AKT 途径来抑制细胞增殖,诱导自噬和凋亡。Actein 在体内几乎没有毒性。
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GC19019
Acumapimod
Acumapimod (BCT197) is an orally active p38 MAP kinase inhibitor, with an IC50 of less than 1 uM for p38α.
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GC32797
AD80
AD80是多种激酶的抑制剂,抑制RET,RAF,SRC和S6K活性,但对mTOR的活性明显减弱。
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GC10204
AEG 3482
inhibitor of Jun kinase (JNK)-dependent apoptosis
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GC17265
AG-126
ERK1 (p44) and ERK2 (p42) inhibitor
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GC12646
AL 8697
p38α inhibitor,potent and selective
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GC14899
AMG 548
P38α inhibitor,potent and selective
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GC38518
AMG-548 dihydrochloride
AMG-548 dihydrochloride 是一种有效的,口服有效的,选择性 p38α 抑制剂 (Ki=0.5 nM),对 p38β 略有选择性 (Ki=36 nM) 并且对 p38γ 和 p38δ 具有 >1000 倍的选择性。AMG-548 dihydrochloride 也有效抑制全血 LPS 刺激的 TNFα (IC50=3 nM)。AMG-548 dihydrochloride 通过直接抑制酪蛋白激酶 1 (Casein kinase 1) 同种型 δ 和 ε 来抑制 Wnt 信号传导。
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GC11559
Anisomycin
JNK agonist, potent and specific
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GC15240
APS-2-79
KSR-dependent MAPK modulator
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GC32692
APTO-253 (LOR-253)
APTO-253是一种Kruppel-likefactor4诱导剂,同时可稳定Gquadruplex结构,具有抗癌活性。
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GN10063
Arctigenin
Anti-inflammatory, antiproliferative
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GC12882
AS 602801
Jun Kinase Inhibitor
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GC10010
AS601245
c-Jun NH2-terminal protein kinase inhibitor