JAK/STAT Signaling

Products for JAK/STAT Signaling
- Cat.No. Product Name Information
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GC38006
β-Hydroxyisovalerylshikonin
Beta-hydroxyisovalerylshikonin 是一种从Lithospermium radix 中分离出的天然产物,是一种有效的 PTK 抑制剂, 对 EGFR 和 v-Src 受体作用的 IC50 分别为 0.7 μM 和 1 μM。Beta-hydroxyisovalerylshikonin 对多种肿瘤细胞系均有抑制作用,能高效诱导 NCI-H522 和 DMS114 细胞的死亡。
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GC34964
(1S,3R,5R)-PIM447 dihydrochloride
(1S,3R,5R)-PIM447 (dihydrochloride)是PIM的抑制剂,来自专利US 20100056576 A1化合物实例72。对Pim1,Pim2和Pim3的IC50分别为0.095,0.522和0.369 μM。
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GC34971
(3R,4S)-Tofacitinib
Tofacitinib(CP-690550)是高效JAK3抑制剂,IC50为1 nM,比对JAK2和JAK1的抑制性高20倍和100倍。
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GC34972
(3S,4R)-Tofacitinib
Tofacitinib(CP-690550)是高效JAK3抑制剂,IC50为1 nM,比对JAK2和JAK1的抑制性高20倍和100倍。
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GC34973
(3S,4S)-Tofacitinib
Tofacitinib(CP-690550)是高效JAK3抑制剂,IC50为1 nM,比对JAK2和JAK1的抑制性高20倍和100倍。
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GC17055
1,2,3,4,5,6-Hexabromocyclohexane
JAK2 tyrosine kinase inhibitor
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GC12138
5,15-DPP
STAT3 inhibitor
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GC32023
Abrocitinib (PF-04965842)
Abrocitinib(PF-04965842)是一种有效、可口服、选择性的JAK1抑制剂,对JAK1和JAK2的IC50值分别为29和803nM。Abrocitinib(PF-04965842)可抑制TYK2的活性(IC50,1.253μM)和刺激后STAT1,STAT3和STAT5的磷酸化水平。可用于自身免疫症的研究。
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GC13257
AC480 (BMS-599626)
HER1/2 inhibitor,selective and efficacious
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GC11892
AEE788 (NVP-AEE788)
EGFR/HER-2/VEGFR inhibitor
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GC10707
Afatinib dimaleate
EGFR inhibitor
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GC13296
Afatinib(BIBW2992)
Irreversible EGFR/HER2 inhibitor
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GC11744
AG 555
Potent EGFR-kinase inhibitor
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GC13168
AG 825
Selective ErbB2 inhibitor
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GC14494
AG 99
EGFR inhibitor
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GC17226
AG-1478
EGFR inhibitor,potent and selective
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GC12864
AG-1557
inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase
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GC17647
AG-18
EGFR/PDGFR inhibitor
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GC13854
AG-490 (Tyrphostin B42)
STAT3/EGFR/JAK2/JAK3 inhibitor
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GN10705
Alantolactone
Extracted from Inula helenium L. roots,Inula grandis chrenk leaves;Store the product in sealed, cool and dry condition