NMDA Receptor(NMDA受体)
NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.
Products for NMDA Receptor
- Cat.No. 产品名称 Information
- GC11124 Lanicemine A low-trapping NMDA channel blocker
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GC11025
(+)-MK 801 Maleate
An NMDA receptor antagonist
- GC16315 D-AP5 A selective NMDA antagonist
- GC11862 LY 233053 Competitive NMDA receptor antagonist
- GC16776 QNZ 46 An antagonist of NR2C- and NR2D-subunit containing NMDA receptors
- GC10085 DQP 1105 An NMDA receptor antagonist
- GC14770 TCN 213 TCN 213 是一种选择性的、可克服的、依赖甘氨酸的 GluN1/GluN2A NMDAR 拮抗剂,在 75、750、7500 nM 甘氨酸存在下,IC50 分别为 0.55、3.5、40 μM。
- GC15065 TCN 201 An NR2A-selective NMDA receptor antagonist
- GC10247 PPDA PPDA 是一种亚型选择性 NMDA 受体拮抗剂,它优先与含有 NR2C/NR2D 的受体结合。
- GC10688 MNI-caged-D-aspartate Agonist at NMDA receptors and EAAT substrate
- GC10574 Norketamine hydrochloride Major metabolite of ketamine, NMDA receptor antagonist
- GC14414 CIQ A subunit-selective NMDA receptor potentiator
- GC14598 5,7-Dichlorokynurenic acid sodium salt An NMDA receptor antagonist
- GC14897 DL-AP5 Sodium salt A competitive NMDA antagonist
- GC14381 Ro 8-4304 hydrochloride NMDA receptor antagonist
- GC10595 threo Ifenprodil hemitartrate σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist
- GC14442 TCS 46b NR1A/NR2B NMDA receptor antagonist,orally active
- GC10792 Co 101244 hydrochloride Co 101244 (PD 174494) hydrochloride 是一种含有 NR2B 的 NMDA 受体拮抗剂。
- GC17481 Gavestinel An NMDA receptor antagonist
- GC11879 PPPA PPPA 是一种竞争性 NMDA 受体拮抗剂,对含 NR2A 的受体具有中等选择性。
- GC14357 PMPA (NMDA antagonist) PMPA(NMDA 拮抗剂)是一种 NMDA 受体拮抗剂,对 NR2A、NR2B、NR2C 和 NR2D 的 Ki 值分别为 0.84、2.74、3.53 和 4.16 μM。
- GC11281 N20C hydrochloride NMDA receptor antagonist
- GC15343 Eliprodil An NMDA receptor antagonist
- GC14782 Ro 04-5595 hydrochloride NR2B-containing NMDA receptors antagonist
- GC16131 Remacemide hydrochloride Remacemide hydrochloride (FPL 12924AA) 是 Na+ 通道的中度抑制剂,是一种弱的非竞争性 NMDA 受体拮抗剂,对 MK-801 结合和 NMDA 电流的 IC50 分别为 68 μM 和 76 μM。
- GC15752 CGP 78608 hydrochloride CGP 78608 hydrochloride 是一种高效的选择性拮抗剂,作用于 NMDA 受体的甘氨酸结合位点,IC50 为 6 nM。
- GC10122 CGP 37849 CGP 37849 是一种有效的、竞争性的和具有口服活性的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂。
- GC11027 CGP 39551 CGP 39551 是一种有效的、具有口服活性的竞争性 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂,具有有效的抗惊厥活性。
-
GC12816
SDZ 220-040
NMDA receptor antagonist
- GC16272 CGS 19755 NMDA receptor antagonist
- GC12137 CCMQ inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites
- GC12873 LY 235959 NMDA receptor antagonist
- GC14810 L-701,324 An NMDA receptor antagonist
- GC10696 L-689,560 L-689,560 是一种有效的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂,作用于 GluN1 甘氨酸结合位点。
- GC11706 L-701,252 L-701,252 是一种有效的甘氨酸位点 NMDA 受体拮抗剂,IC50 为 420 nM。
- GC15732 Synthalin sulfate NMDA receptor antagonist
- GC10471 Ifenprodil hemitartrate An NMDA receptor antagonist
- GC10237 (±)-1-(1,2-Diphenylethyl)piperidine maleate NMDA receptor antagonist
- GC10168 (R)-4-Carboxyphenylglycine NMDA receptor antagonist
- GC12488 (RS)-(Tetrazol-5-yl)glycine An NMDA receptor agonist
- GC16799 5,7-Dichlorokynurenic acid An NMDA receptor antagonist
- GC10370 (S)-(-)-HA-966 (S)-(-)-HA-966 ((-)-HA 966) 是一种 γ-Hydroxybutyrate 样剂,作为 NMDA 受体拮抗剂的活性较弱。
- GC14085 (R)-(+)-HA-966 (R)-(+)-HA-966 ((+)-HA-966) 是 N-甲基-D-天冬氨酸 (NMDA) 受体复合物甘氨酸位点的部分激动剂/拮抗剂。
- GC14236 (R)-CPP An NMDA receptor antagonist
- GC10114 Homoquinolinic acid NMDA receptor agonist
- GC11942 cis-ACPD cis-ACPD 是一种有效的 NMDA 受体激动剂,IC50 为 3.3 μM。
- GC10476 (RS)-CPP NMDA antagonist
- GC15112 D-AP7 NMDA receptor antagonist
- GC12154 L-AP5 NMDA拮抗剂
- GC17206 DL-AP5 A competitive NMDA antagonist