GPCR/G protein - Signaling Pathways

Cat.No. Product Name Information

GC38007 β-Melanocyte Stimulating Hormone (MSH), human TFA β-Melanocyte Stimulating Hormone (MSH), human TFA, 是一个 22 肽，是一种内源性黑皮质素-4 受体 (melanocortin-4 receptor; MC4-R) 激动剂。

GC37983 β3-AR agonist 1 β3-AR agonist 1 (compound 15) 是一种高效选择性的，可口服的 β3-肾上腺素能受体 (β3-AR) 激动剂 (EC50=18 nM)，对 β1-、β2-、α1A-AR 无活性 (β1/β3, β2/β3, α1A/β3>556倍)。

GC17002 γ1-MSH melanocortin MC3 receptor agonist

GC15519 α-CGRP (human) Endogenous calcitonin gene-related peptide receptor (CGRP) agonist

GC11346 α-helical CRF 9-41 Antagonist of corticotropin releasing factor receptor

GC11577 α-Methyl-5-hydroxytryptamine maleate 5-HT2B receptor agonist

GC14374 α-MSH Endogenous melanocortin receptor agonist

GC31237 α1 adrenoceptor-MO-1 α1adrenoceptor-MO-1是一种S型对映体，对alpha1adrenergicreceptor具有亲和性，可以抗α-肾上腺素能，同时能够止痛；比R型对映体的活性高。

GC33681 β-Caryophyllene ((−)-trans-Caryophyllene) β-Caryophyllene是一个CB2受体激动剂。

GC33693 β-Melanocyte Stimulating Hormone (MSH), human (Beta-MSH (1-22) (human)) β-MelanocyteStimulatingHormone(MSH),human是黑皮质素受体(melanocortin(MC)receptor)激动剂。

GC31573 β3-AR agonist 2 β3-ARagonist2是一种有效的选择性β3肾上腺素能受体(β3-adrenergicreceptor，β3-AR)激动剂，EC50为8nM。

GC34231 γ-1-Melanocyte Stimulating Hormone (MSH), amide γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。