GPCR/G protein
- Neuropeptide FF/AF Receptors(32)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(381)
- Acetylcholine(3)
- Adenosine Deaminase(6)
- Adenosine Receptor(104)
- Adenosine Kinase(3)
- Adiponectin Receptor(3)
- Adrenergic Receptor(290)
- Adrenergic Transporters(5)
- Apelin Receptor(7)
- Angiotensin Receptor(74)
- Bombesin Receptors(19)
- Bradykinin Receptors(22)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(112)
- Calcimimetic Agent(2)
- CaSR(16)
- CCK1 Receptors(6)
- CCK2 Receptors(7)
- CCR(47)
- Chemokine Receptors(19)
- CRF1 Receptors(8)
- CRF2 Receptors(3)
- CXCR(54)
- CysLT1 receptor(1)
- Endothelin Receptor(38)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(13)
- Galanin Receptors(11)
- Ghrelin Receptors(10)
- GHSR(15)
- GIP Receptor(2)
- Glucagon Receptor(49)
- Glucocorticoid Receptor(65)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(11)
- GPR109A(3)
- GPR119(9)
- GPR120(9)
- GPR35(7)
- GPR44(1)
- GPR55(8)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(47)
- LPA Receptor(12)
- LPL Receptor(39)
- LTD4 Receptor(1)
- mGluR (69)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(35)
- Melatonin Receptors(18)
- Motilin Receptor(6)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(11)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(21)
- NPY Receptors(24)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(28)
- Oxytocin Receptors(18)
- P2Y Receptor(43)
- PACAP Receptors(3)
- PAF Receptors(8)
- Peptide Receptors(8)
- PGD2 Receptor(1)
- Prostaglandin Receptor(110)
- Protease-Activated Receptors(10)
- Prostanoid Receptors(25)
- RGS(2)
- S1P receptor(6)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(26)
- Sigma Receptor(42)
- Vasopressin Receptor(18)
- 17,20-lyase(3)
- Ras(64)
- Urotensin-II Receptor(10)
- VIP Receptors(7)
- EBI2/GPR183(4)
- TSH Receptor(4)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(3)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(4)
- CRFR(16)
- RGS Protein(4)
- Urotensin Receptor(1)
- Cholecystokinin Receptor(22)
- GPR139(1)
- mAChR(124)
- MCHR1 (GPR24)(14)
- Neurokinin Receptor(55)
- Cat.No. Product Name Information
-
GC38007
β-Melanocyte Stimulating Hormone (MSH), human TFA
β-Melanocyte Stimulating Hormone (MSH), human TFA, 是一个 22 肽,是一种内源性黑皮质素-4 受体 (melanocortin-4 receptor; MC4-R) 激动剂。
-
GC37983
β3-AR agonist 1
β3-AR agonist 1 (compound 15) 是一种高效选择性的,可口服的 β3-肾上腺素能受体 (β3-AR) 激动剂 (EC50=18 nM),对 β1-、β2-、α1A-AR 无活性 (β1/β3, β2/β3, α1A/β3>556倍)。
-
GC17002
γ1-MSH
melanocortin MC3 receptor agonist
-
GC15519
α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist
-
GC11346
α-helical CRF 9-41
Antagonist of corticotropin releasing factor receptor
-
GC11577
α-Methyl-5-hydroxytryptamine maleate
5-HT2B receptor agonist
-
GC14374
α-MSH
Endogenous melanocortin receptor agonist
-
GC31237
α1 adrenoceptor-MO-1
α1adrenoceptor-MO-1是一种S型对映体,对alpha1adrenergicreceptor具有亲和性,可以抗α-肾上腺素能,同时能够止痛;比R型对映体的活性高。
-
GC33681
β-Caryophyllene ((−)-trans-Caryophyllene)
β-Caryophyllene是一个CB2受体激动剂。
-
GC33693
β-Melanocyte Stimulating Hormone (MSH), human (Beta-MSH (1-22) (human))
β-MelanocyteStimulatingHormone(MSH),human是黑皮质素受体(melanocortin(MC)receptor)激动剂。
-
GC31573
β3-AR agonist 2
β3-ARagonist2是一种有效的选择性β3肾上腺素能受体(β3-adrenergicreceptor,β3-AR)激动剂,EC50为8nM。
-
GC34231
γ-1-Melanocyte Stimulating Hormone (MSH), amide
γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。
-
GC17413
(±)-5'-Chloro-5'-deoxy-ENBA
adenosine A1 receptor agonist, selective and high-affinity
-
GC17408
(±)-AC 7954 hydrochloride
urotensin-II (UT) receptor agonist
-
GC15045
(±)-AMG 487
CXCR3 antagonist
-
GC16838
(±)-Cloprostenol sodium salt
prostaglandin F2α (PGF2α) analog,FP receptor agonist
-
GC18090
(±)-J 113397
NOP receptor antagonist
-
GC15144
(±)-PPCC oxalate
sigma (σ) receptor ligand
-
GC10907
(±)-SLV 319
CB1 receptor antagonist,potent and selective
-
GC12394
(±)-trans-ACPD
metabotropic glutamate receptors agonist