GPCR/G protein
- Neuropeptide FF/AF Receptors(39)
- Formyl Peptide Receptors(11)
- 5-HT Receptor(431)
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- Adrenergic Transporters(5)
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- Angiotensin Receptor(92)
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- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(124)
- Calcimimetic Agent(2)
- CaSR(17)
- CCK1 Receptors(8)
- CCK2 Receptors(7)
- CCR(54)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
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- CXCR(57)
- CysLT1 receptor(1)
- Endothelin Receptor(44)
- EP1 Receptor(2)
- EP4 Receptor(3)
- ERRγ(1)
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- GHSR(18)
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- Glucagon Receptor(58)
- Glucocorticoid Receptor(74)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(3)
- GPR119(10)
- GPR120(9)
- GPR35(7)
- GPR44(1)
- GPR55(9)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(51)
- LPA Receptor(12)
- LPL Receptor(42)
- LTD4 Receptor(1)
- mGluR (90)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(39)
- Melatonin Receptors(19)
- Motilin Receptor(6)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(17)
- NK2 Receptors(7)
- NK3 Receptor(6)
- NOP Receptor(21)
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- Orexin(3)
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- OX Receptor(32)
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- P2Y Receptor(52)
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- PGD2 Receptor(1)
- Prostaglandin Receptor(145)
- Protease-Activated Receptors(10)
- RGS(2)
- S1P receptor(8)
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- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(28)
- Sigma Receptor(48)
- Vasopressin Receptor(28)
- 17,20-lyase(5)
- Ras(72)
- Urotensin-II Receptor(11)
- VIP Receptors(7)
- EBI2/GPR183(4)
- TSH Receptor(5)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(21)
- GPR84(3)
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- Kisspeptin Receptor(4)
- CRFR(19)
- RGS Protein(5)
- Urotensin Receptor(5)
- Cholecystokinin Receptor(24)
- GPR139(1)
- mAChR(147)
- MCHR1 (GPR24)(15)
- Neurokinin Receptor(62)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(12)
- GRK(1)
- Cat.No. Product Name Information
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GC38007
β-Melanocyte Stimulating Hormone (MSH), human TFA
β-Melanocyte Stimulating Hormone (MSH), human TFA, 是一个 22 肽，是一种内源性黑皮质素-4 受体 (melanocortin-4 receptor; MC4-R) 激动剂。
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GC37983
β3-AR agonist 1
β3-AR agonist 1 (compound 15) 是一种高效选择性的，可口服的 β3-肾上腺素能受体 (β3-AR) 激动剂 (EC50=18 nM)，对 β1-、β2-、α1A-AR 无活性 (β1/β3, β2/β3, α1A/β3>556倍)。
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GC40105
βARK1 Inhibitor
βARK1 inhibitor is an inhibitor of G protein-coupled receptor kinase 2/β-adrenergic receptor kinase 1 (GRK2/βARK1; IC50 = 126 μM).
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GC61462
γ-1-Melanocyte Stimulating Hormone (MSH), amide
γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。
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GC17002
γ1-MSH
melanocortin MC3 receptor agonist
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GC15519
α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist
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GC11346
α-helical CRF 9-41
Antagonist of corticotropin releasing factor receptor
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GC11577
α-Methyl-5-hydroxytryptamine maleate
5-HT2B receptor agonist
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GC31237
α1 adrenoceptor-MO-1
α1adrenoceptor-MO-1是一种S型对映体，对alpha1adrenergicreceptor具有亲和性，可以抗α-肾上腺素能，同时能够止痛；比R型对映体的活性高。
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GC33681
β-Caryophyllene ((−)-trans-Caryophyllene)
β-Caryophyllene是一个CB2受体激动剂。
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GC33693
β-Melanocyte Stimulating Hormone (MSH), human (Beta-MSH (1-22) (human))
β-MelanocyteStimulatingHormone(MSH),human是黑皮质素受体(melanocortin(MC)receptor)激动剂。
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GC31573
β3-AR agonist 2
β3-ARagonist2是一种有效的选择性β3肾上腺素能受体(β3-adrenergicreceptor，β3-AR)激动剂，EC50为8nM。
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GC34231
γ-1-Melanocyte Stimulating Hormone (MSH), amide
γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。
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GC17413
(±)-5'-Chloro-5'-deoxy-ENBA
adenosine A1 receptor agonist, selective and high-affinity
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GC17408
(±)-AC 7954 hydrochloride
urotensin-II (UT) receptor agonist
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GC15045
(±)-AMG 487
CXCR3 antagonist
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GC41668
(±)-Clopidogrel (hydrochloride)
Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM).
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GC16838
(±)-Cloprostenol sodium salt
prostaglandin F2α (PGF2α) analog,FP receptor agonist
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GC46283
(±)-Clorprenaline-d7
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GC18090
(±)-J 113397
NOP receptor antagonist
