GPCR/G protein
- Neuropeptide FF/AF Receptors(39)
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- mGluR (93)
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- GPR81(1)
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- GPR139(1)
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- Neurokinin Receptor(65)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(16)
- GRK(1)
- Cat.No. Product Name Information
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GC38007
β-Melanocyte Stimulating Hormone (MSH), human TFA
β-Melanocyte Stimulating Hormone (MSH), human TFA, 是一个 22 肽，是一种内源性黑皮质素-4 受体 (melanocortin-4 receptor; MC4-R) 激动剂。
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GC37983
β3-AR agonist 1
β3-AR agonist 1 (compound 15) 是一种高效选择性的，可口服的 β3-肾上腺素能受体 (β3-AR) 激动剂 (EC50=18 nM)，对 β1-、β2-、α1A-AR 无活性 (β1/β3, β2/β3, α1A/β3>556倍)。
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GC40105
βARK1 Inhibitor
βARK1 inhibitor is an inhibitor of G protein-coupled receptor kinase 2/β-adrenergic receptor kinase 1 (GRK2/βARK1; IC50 = 126 μM).
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GC61462
γ-1-Melanocyte Stimulating Hormone (MSH), amide
γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。
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GC17002
γ1-MSH
melanocortin MC3 receptor agonist
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GC62708
σ1 Receptor antagonist-1
σ1 Receptor antagonist-1 是一种高效且选择性的 sigma 1 受体拮抗剂 (pKi=10.28)。σ1 Receptor antagonist-1 抑制细胞生长，在 G0/G1 期阻滞细胞周期并诱导 MCF-7/ADR 细胞凋亡 (apoptosis)。
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GC15519
α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist
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GC11346
α-helical CRF 9-41
Antagonist of corticotropin releasing factor receptor
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GC11577
α-Methyl-5-hydroxytryptamine maleate
5-HT2B receptor agonist
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GC31237
α1 adrenoceptor-MO-1
α1adrenoceptor-MO-1是一种S型对映体，对alpha1adrenergicreceptor具有亲和性，可以抗α-肾上腺素能，同时能够止痛；比R型对映体的活性高。
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GC33681
β-Caryophyllene ((−)-trans-Caryophyllene)
β-Caryophyllene是一个CB2受体激动剂。
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GC33693
β-Melanocyte Stimulating Hormone (MSH), human (Beta-MSH (1-22) (human))
β-MelanocyteStimulatingHormone(MSH),human是黑皮质素受体(melanocortin(MC)receptor)激动剂。
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GC31573
β3-AR agonist 2
β3-ARagonist2是一种有效的选择性β3肾上腺素能受体(β3-adrenergicreceptor，β3-AR)激动剂，EC50为8nM。
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GC34231
γ-1-Melanocyte Stimulating Hormone (MSH), amide
γ-1-MelanocyteStimulatingHormone(MSH),amide是一种含11个氨基酸的多肽。γ-1-MelanocyteStimulatingHormone通过激活黑皮质素受体3(MC3-R)来调节钠(Na+)平衡和血压。
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GC17413
(±)-5'-Chloro-5'-deoxy-ENBA
adenosine A1 receptor agonist, selective and high-affinity
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GC17408
(±)-AC 7954 hydrochloride
urotensin-II (UT) receptor agonist
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GC15045
(±)-AMG 487
CXCR3 antagonist
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GC41668
(±)-Clopidogrel (hydrochloride)
Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM).
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GC16838
(±)-Cloprostenol sodium salt
prostaglandin F2α (PGF2α) analog,FP receptor agonist
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GC46283
(±)-Clorprenaline-d7
