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Cyproheptadine (hydrochloride hydrate) 目录号 GC43353

An antihistamine with antiserotonergic and anticholinergic activities

规格 价格 库存 购买数量
100mg
¥590.00
现货
250mg
¥1,331.00
现货
500mg
¥2,359.00
现货
1g
¥3,251.00
现货

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Sample solution is provided at 25 µL, 10mM.

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Chemical Properties

Cas No. 41354-29-4 SDF Download SDF
别名 N/A
化学名 N/A
Canonical SMILES CN(CC/1)CCC1=C2C(C=CC=C3)=C3C=CC4=C\2C=CC=C4.CN(CC/5)CCC5=C6C(C=CC=C7)=C7C=CC8=C\6C=CC=C8.Cl.O.O.O.Cl
分子式 C21H21N•HCl [1.5H2O] 分子量 350.9
溶解度 DMF: 30 mg/mL,DMSO: 30 mg/mL,Ethanol: 30 mg/mL,Ethanol:PBS(pH 7.2) (1:1): 0.5 mg/mL 储存条件 Store at -20°C
General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
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产品描述

Cyproheptadine is a first-generation antihistamine that potently antagonizes the histamine H1 receptor (pKi = 9.42). It also antagonizes serotonin and muscarinic receptors at nanomolar concentrations. Cyproheptadine also inhibits the lysine methyltransferase SET7/9 (IC50 = 1 µM), suppressing the expression of estrogen receptor α in human breast cancer MCF-7 cells.